SCHEMBL5487758

SCHEMBL5487758

CCCCCCC[Si](C)(C)CC(N)=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SOAT1 P35610 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
FAAH O00519 1/20 0.42
TP53 P04637 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C19 P33261 1/20 0.42
KDM4E B2RXH2 2/20 0.39
EPHX1 P07099 4/20 0.39
CES2 O00748 3/20 0.38
CES1 P23141 3/20 0.38
PPARG P37231 6/20 0.37
PPARD Q03181 6/20 0.37
PPARA Q07869 6/20 0.37
HDAC11 Q96DB2 5/20 0.37
TSHR P16473 4/20 0.37
GPR84 Q9NQS5 4/20 0.37
ALDH1A1 P00352 2/20 0.37
TLR2 O60603 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5483154 0.98 SOAT1 (0.39) SOAT1MEN1KMT2AFAAHTP53
SCHEMBL537434 0.91 SOAT1 (0.36) SOAT1MEN1KMT2AFAAHTP53
SCHEMBL30701400 0.83 SOAT1 (0.57) SOAT1MEN1KMT2AFAAHTP53
SCHEMBL30701337 0.83 SOAT1 (0.57) SOAT1MEN1KMT2AFAAHTP53
SCHEMBL5487841 0.82 MEN1 (0.30) SOAT1MEN1KMT2AFAAHTP53
SCHEMBL9634443 0.76 FAAH (0.42) MEN1KMT2AFAAHEPHX1CES2
SCHEMBL12296678 0.76 NAAA (0.42) MEN1KMT2AFAAHCYP1A2EPHX1
SCHEMBL10356297 0.74 TSHR (0.53) MEN1KMT2AEPHX1TSHRALDH1A1
SCHEMBL19119178 0.74 TSHR (0.53) MEN1KMT2AEPHX1TSHRALDH1A1
SCHEMBL10356295 0.74 TSHR (0.53) MEN1KMT2AEPHX1TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1737471-A2 PHARMACEUTICAL COMPOSITIONS AND METHODS OF USE OF LIPOPHILIC, SILICON-SUBSTITUTED, CYCLOOXYGENASE-2 SELECTIVE NON-STEROIDAL ANTI-INFLAMMATORY DRUGS AND DERIVATIVES RND Pharmaceuticals (US) 2007-01-03 EP claimed
WO-2005102358-A2 SILICONE-SUBSTITUTED COX-2 SELECTIVE INHIBITORS RND PHARMACEUTICALS (US) 2005-11-03 WO claimed