SCHEMBL5488644

SCHEMBL5488644

CC(C)(C)OC(=O)NCCCC[C@@H](CNCCc1c[nH]c2ccccc12)NC(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.49
TACR1 P25103 3/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HDAC9 Q9UKV0 1/20 0.41
HDAC5 Q9UQL6 1/20 0.41
KMT2A Q03164 1/20 0.41
NMBR P28336 5/20 0.41
CTSL P07711 1/20 0.41
CTSS P25774 1/20 0.41
CTSK P43235 1/20 0.41
FAAH O00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4614285 0.87 NMBR (0.52) PIN1TACR1HDAC3HDAC4HDAC1
SCHEMBL5496357 0.83 PIN1 (0.43) PIN1HDAC3HDAC4HDAC1HDAC7
SCHEMBL18725627 0.82 KMT2A (0.55) KMT2A
SCHEMBL18826572 0.82 KMT2A (0.48) KMT2A
SCHEMBL17935596 0.82 KMT2A (0.55) KMT2A
SCHEMBL4890850 0.81 TACR1 (0.53) TACR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL4890847 0.81 TACR1 (0.53) TACR1HDAC3HDAC4HDAC1HDAC7
SCHEMBL21461837 0.80 KMT2A (0.55) KMT2A
SCHEMBL29400817 0.80 KMT2A (0.53) KMT2A
SCHEMBL2947901 0.80 KMT2A (0.53) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7163921-B1 Peptide derivatives and medicinal compositions NIPPON SHINYAKU CO., LTD. (JP) 2007-01-16 US disclosed
EP-1275657-A1 PEPTIDE DERIVATIVES AND MEDICINAL COMPOSITIONS Nippon Shinyaku Co., Ltd. (JP) 2003-01-15 EP disclosed