SCHEMBL5488918

SCHEMBL5488918

CCOC(=O)c1c(SC)nc2ccccc2c1O.CSc1[nH]c2ccccc2c(=O)c1C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.48
ALDH1A1 P00352 5/20 0.41
MAPT P10636 5/20 0.41
KDM4E B2RXH2 4/20 0.41
LMNA P02545 3/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
MAPK10 P53779 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
TUBB4A P04350 1/20 0.39
TUBB P07437 1/20 0.39
TUBA3C P0DPH7 1/20 0.39
TUBA1B P68363 1/20 0.39
TUBA4A P68366 1/20 0.39
TUBB4B P68371 1/20 0.39
TUBB3 Q13509 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL395812 0.84 SMN1; SMN2 (0.53) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL397184 0.77 KDM4E (0.53) RXFP1ALDH1A1MAPTKDM4ELMNA
SCHEMBL14472396 0.74 KDM4E (0.63) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL10257067 0.73 CYP2D6 (0.52) MAPTLMNAKMT2AMEN1TDP1
SCHEMBL11075264 0.70 KDM4E (0.61) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL6300719 0.70 ALDH1A1 (0.67) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL29860485 0.70 SMN1; SMN2 (0.58) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL19846945 0.70 KDM4E (0.58) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL27659536 0.70 SMN1; SMN2 (0.58) ALDH1A1MAPTKDM4ELMNAKMT2A
SCHEMBL538291 0.70 SMN1; SMN2 (0.69) ALDH1A1MAPTKDM4ELMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2502913-A2 Modulators of ATP-binding cassette transporters Vertex Pharmaceuticals Incorporated (US) 2012-09-26 EP disclosed
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed