SCHEMBL5489033

SCHEMBL5489033

Cc1c(Cl)ccc2c1NC(=O)C2(c1ccc(O)cc1)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.48
CNR1 P21554 1/20 0.48
GPR35 Q9HC97 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
MMP2 P08253 1/20 0.46
MMP13 P45452 1/20 0.46
LMNA P02545 3/20 0.46
CYP1A2 P05177 1/20 0.46
PTGS1 P23219 1/20 0.46
SLC6A2 P23975 1/20 0.46
CYP2C19 P33261 1/20 0.46
PTGS2 P35354 1/20 0.46
SLC6A3 Q01959 1/20 0.46
HIF1A Q16665 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CHRM2 P08172 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
KCNH2 Q12809 1/20 0.41
MAOB P27338 2/20 0.38
MEN1 O00255 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8279032 0.85 MMP2 (0.48) MMP2MMP13LMNACYP1A2PTGS1
SCHEMBL5474643 0.84 CNR1 (0.61) HTTCNR1GPR35GPR55MMP2
SCHEMBL5485571 0.83 CNR1 (0.52) HTTCNR1GPR35GPR55CHRM2
SCHEMBL5479452 0.81 LMNA (0.48) HTTCNR1GPR35GPR55MMP2
SCHEMBL5474437 0.81 CNR1 (0.57) HTTCNR1GPR35GPR55MMP2
SCHEMBL22111762 0.80 CNR1 (0.48) HTTCNR1GPR35GPR55MMP2
SCHEMBL22111806 0.80 CNR1 (0.48) HTTCNR1GPR35GPR55MMP2
SCHEMBL22076805 0.80 CNR1 (0.48) HTTCNR1GPR35GPR55MMP2
SCHEMBL5482053 0.75 MAPT (0.56) HTTCNR1GPR35GPR55LMNA
SCHEMBL5478235 0.74 HTT (0.46) HTTCNR1GPR35GPR55LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070299102-A1 Diphenyl Ox-Indol-2-One Compounds and Their Use in the Treatment of Cancer TOPO TARGET A/S (DK) 2007-12-27 US disclosed
EP-1734951-A2 DIPHENYL-INDOL-2-ON COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER TopoTarget A/S (DK) 2006-12-27 EP disclosed
WO-2005097107-A2 DIPHENYL - INDOL-2-ON COMPOUNDS AND THEIR USE IN THE TREATMENT OF CANCER TOPOTARGET A/S (DK) 2005-10-20 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070299102-A1 Diphenyl Ox-Indol-2-One Compounds and Their Use in the Treatment of Cancer MTOR, RICTOR, CDK4 HTT 1880/4885CNR1 973/4885GPR35 2558/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.