SCHEMBL5489358

SCHEMBL5489358

CC(CN)Cc1nc2cnccc2c(=O)n1Cc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.48
PDE4B Q07343 2/20 0.48
PDE4C Q08493 2/20 0.48
PDE4D Q08499 2/20 0.48
ALDH1A1 P00352 7/20 0.43
KMT2A Q03164 2/20 0.43
KDM4E B2RXH2 2/20 0.43
RAD1 O60671 1/20 0.43
MAPT P10636 1/20 0.43
CFTR P13569 1/20 0.43
APEX1 P27695 1/20 0.43
CASP6 P55212 1/20 0.43
RAD51 Q06609 1/20 0.43
HKDC1 Q2TB90 1/20 0.43
GOPC Q9HD26 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RAB9A P51151 2/20 0.43
POLB P06746 1/20 0.43
LMNA P02545 4/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4314434 0.89 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL5759177 0.83 KIF11 (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL5604490 0.83 KIF11 (0.54) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL5111971 0.81 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL6518180 0.81 PDE4A (0.66) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL5486903 0.81 KIF11 (0.51) ALDH1A1KMT2AKDM4ECYP2C19SMN1; SMN2
SCHEMBL5489353 0.78 ALDH1A1 (0.45) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL13577682 0.77 ALDH1A1 (0.47) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL4320409 0.76 ALDH1A1 (0.45) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL5489055 0.75 KIF11 (0.47) PDE4APDE4BPDE4CPDE4DALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1855664-A2 MITOTIC KINESIN INHIBITORS Merck & Co., Inc. (US) 2007-11-21 EP disclosed
WO-2006078575-A2 FLUORINATED AMINOALKYL-4-OXO-3,4-DIHYDROPYRIDO[3,4- D] PYRIMIDINES AS INHIBITORS OF MITOTIC KINESINS MERCK & CO., INC. (US) 2006-07-27 WO disclosed