P-Toluenesulfonamide

P-Toluenesulfonamide

SCHEMBL5492056

Cc1ccc(S(N)(=O)=O)cc1.[KH]

nearest known ligand 0.95

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 11/20 0.95
CA9 Q16790 10/20 0.95
CA12 O43570 9/20 0.95
CA1 P00915 8/20 0.95
CA7 P43166 4/20 0.95
CA6 P23280 3/20 0.95
CA5A P35218 3/20 0.95
CA5B Q9Y2D0 3/20 0.95
CA3 P07451 2/20 0.95
PTPN7 P35236 1/20 0.62
PTGS2 P35354 5/20 0.60
PTGS1 P23219 2/20 0.60
GAA P10253 1/20 0.59
CA4 P22748 3/20 0.58
CA13 Q8N1Q1 2/20 0.56
CA14 Q9ULX7 2/20 0.56
USP2 O75604 1/20 0.56
TSHR P16473 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
AGO2 Q9UKV8 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
P-Toluenesulfonamide SCHEMBL1331323 0.97 CA2 (1.00) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL31527821 0.97 CA2 (1.00) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL7370 0.97 CA2 (1.00) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL9377640 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL8070437 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL8071454 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL357964 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL8376384 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL15401330 0.95 CA2 (0.95) CA2CA9CA12CA1CA7
P-Toluenesulfonamide SCHEMBL391243 0.95 CA2 (0.95) CA2CA9CA12CA1CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0211944-B1 CARBONATE POLYMER COMPOSITIONS CONTAINING A SALT OF AN AROMATIC SULFONAMIDE AND A FREE AROMATIC SULFIMIDE THE DOW CHEMICAL COMPANY (US) 1989-08-16 EP claimed
CN-113754509-A Method for preparing conjugated diene with single stereo configuration from allyl alcohol compound 中山大学 2021-12-07 CN disclosed
EP-2484725-B1 POLYESTER RESIN COMPOSITION, POLYESTER FIBER, POLYESTER RESIN MOLDED ARTICLE, AND PROCESS FOR PRODUCTION OF NUCLEATING AGENT FOR POLYESTER RESIN ADEKA CORP (JP) 2017-07-19 EP disclosed
US-20140001672-A1 POLYESTER RESIN COMPOSITION, POLYESTER FIBER, POLYESTER RESIN MOLDED ARTICLE, AND PROCESS FOR PRODUCTION OF NUCLEATING AGENT FOR POLYESTER RESIN ADEKA CORPORATION (JP) 2014-01-02 US disclosed
EP-1137642-B1 BIS-SULFONAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2007-12-05 EP disclosed
CN-1332942-C Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists ACTELION PHARMACEUTICALS LTD (CH) 2007-08-22 CN disclosed
US-20060079533-A1 Methods of treating alzheimer's disease NIEMAN JAMES A 2006-04-13 US disclosed
CN-1703397-A Sulfonylamino-acetic acid derivatives and their use as orexin receptor antagonists ACTELION PHARMACEUTICALS LTD (CH) 2005-11-30 CN disclosed
US-6596719-B1 Manufacturing those compounds, pharmaceutical compositions containing one or more of those compounds as endothelin antagonists, and a method of treating a subject having a disorder involving endothelin with the compounds of the ACTELIO PHARMACEUTICALS LTD. (CH) 2003-07-22 US disclosed
WO-2002076440-A2 METHODS OF TREATING ALZHEIMER'S DISEASE WITH PIPERIDIN DERIVATES ELAN PHARMACEUTICALS, INC. (US) 2002-10-03 WO disclosed
WO-2001017976-A1 BIS-SULFONAMIDES ACTELION PHARMACEUTICALS LTD (CH) 2001-03-15 WO disclosed
US-6150526-A Piperidine derivative having renin inhibiting activity HOFFMANN-LA ROCHE INC. (US) 2000-11-21 US disclosed
US-6051712-A PREVENTION OF HIGH BLOOD PRESSURE AND CARDIAC INSUFFICIENCY, AS WELL AS GLAUCOMA, CARDIAC INFARCT, KIDNEY INSUFFICIENCY AND RESTENOSIS HOFFMANN-LA ROCHE INC. (US) 2000-04-18 US disclosed
US-5270313-A Treatment of circulatory disorders HOFFMANN-LA ROCHE INC. (US) 1993-12-14 US disclosed
EP-0211944-B1 CARBONATE POLYMER COMPOSITIONS CONTAINING A SALT OF AN AROMATIC SULFONAMIDE AND A FREE AROMATIC SULFIMIDE THE DOW CHEMICAL COMPANY (US) 1989-08-16 EP disclosed
US-4300897-A SAFE FOR DYED FABRICS; ALSO CONTAINS AN AROMATIC SULFONAMIDE COLGATE-PALMOLIVE COMPANY (US) 1981-11-17 US disclosed
US-4183955-A Troponyl-oxamic acid derivatives for treating allergic conditions Ayerst. McKenna & Harrison Limited (CA) 1980-01-15 US disclosed
US-4125625-A ANTIALLERGENS AYERST, MCKENNA & HARRISON LIMITED (CA) 1978-11-14 US disclosed
US-4123376-A AROMATIC SULFONAMIDE COLGATE-PALMOLIVE COMPANY (US) 1978-10-31 US disclosed
US-4057556-A ANTIALLERGENS AYERST, MCKENNA & HARRISON LTD. (CA) 1977-11-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060079533-A1 Methods of treating alzheimer's disease BACE1, PSEN1, PSEN2 CA2 1585/4885CA9 3420/4885CA12 2820/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.