SCHEMBL5492322

SCHEMBL5492322

Nc1cc(O)c(C2C3CC4CC(C3)CC2C4)cc1F.Nc1cc(O)c(C2C3CC4CC(C3)CC2C4)cc1F

nearest known ligand 0.31

Predicted protein targets (top 1)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL435480 1.00 SCN9A (0.30) SCN9A
SCHEMBL436183 0.79 CYP3A4 (0.34) SCN9A
SCHEMBL4614199 0.79 SCN9A (0.35) SCN9A
SCHEMBL16046506 0.69 CHRNB2 (0.38) SCN9A
SCHEMBL22321085 0.68 MEN1 (0.41) SCN9A
SCHEMBL27199191 0.68 CNR1 (0.37) SCN9A
SCHEMBL5492318 0.68 MEN1 (0.41)
SCHEMBL435479 0.68 MEN1 (0.41)
SCHEMBL7167055 0.67 TAAR1 (0.32)
SCHEMBL8795608 0.67 SCN9A (0.36) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed