SCHEMBL5492849

SCHEMBL5492849

O=C(NO)c1ccc(C#CCNC(=O)c2cc3cc(OCCN4CCCC4)ccc3o2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 4/20 0.46
HDAC6 Q9UBN7 2/20 0.46
JAK2 O60674 1/20 0.46
BRD4 O60885 1/20 0.46
RET P07949 1/20 0.46
JAK1 P23458 1/20 0.46
TYK2 P29597 1/20 0.46
FLT3 P36888 1/20 0.46
JAK3 P52333 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
ADAM17 P78536 5/20 0.45
MCHR1 Q99705 1/20 0.44
KDM4E B2RXH2 1/20 0.44
KDM1A O60341 1/20 0.44
HDAC3 O15379 1/20 0.44
HTR6 P50406 1/20 0.44
HDAC2 Q92769 1/20 0.44
NCOR2 Q9Y618 1/20 0.44
ACACB O00763 2/20 0.43
PSMB1 P20618 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4817770 0.99 HDAC1 (0.46) HDAC1HDAC6JAK2BRD4RET
SCHEMBL5498703 0.94 HDAC1 (0.52) HDAC1HDAC6HDAC8KDM4EKDM1A
SCHEMBL4247487 0.93 ADAM17 (0.44) HDAC1HDAC6JAK2BRD4RET
Hydrochloric Acid SCHEMBL4809157 0.93 HDAC1 (0.51) HDAC1HDAC6HDAC8KDM4EKDM1A
SCHEMBL416282 0.88 HPGD (0.51) HDAC1HDAC6JAK2BRD4RET
SCHEMBL4816497 0.87 HDAC3 (0.46) HDAC1HDAC6HDAC8HDAC3HDAC2
SCHEMBL4253905 0.86 ALDH1A1 (0.45) HDAC1KDM4EKDM1AACACBPSMB1
SCHEMBL447779 0.86 HDAC1 (0.50) HDAC1HDAC6JAK2BRD4RET
Hydrochloric Acid SCHEMBL5970288 0.84 CHEK2 (0.40) HDAC1HDAC6HDAC8HDAC3HDAC2
SCHEMBL444969 0.83 ADAM17 (0.45) HDAC1HDAC6JAK2BRD4RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1656348-B1 ACETYLENE DERIVATIVES AS INHIBITORS OF HISTONE DEACETYLASE AXYS PHARM INC (US) 2007-02-07 EP claimed