Naptalam

Naptalam

SCHEMBL54940

O=C(O)c1ccccc1C(=O)Nc1cccc2ccccc12

nearest known ligand 0.74

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.74
CHRNB2 P17787 1/20 0.70
CHRNB4 P30926 1/20 0.70
CHRNA3 P32297 1/20 0.70
CHRNA4 P43681 1/20 0.70
NPC1 O15118 3/20 0.69
RAB9A P51151 3/20 0.69
CYP1A2 P05177 1/20 0.68
CYP3A4 P08684 1/20 0.68
CYP2D6 P10635 1/20 0.68
CYP2C9 P11712 1/20 0.68
CYP2C19 P33261 1/20 0.68
GFER P55789 1/20 0.62
KMT2A Q03164 3/20 0.60
ALDH1A1 P00352 3/20 0.60
GAA P10253 2/20 0.60
MEN1 O00255 2/20 0.60
SMN1; SMN2 Q16637 2/20 0.60
TP53 P04637 1/20 0.60
NFKB1 P19838 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Naptalam SCHEMBL29610802 1.00 HSD17B10 (0.74) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
Naptalam SCHEMBL29469565 1.00 HSD17B10 (0.74) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
Naptalam SCHEMBL8537412 1.00 HSD17B10 (0.74) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
Naptalam SCHEMBL984498 0.98 HSD17B10 (0.72) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL13927141 0.91 HSD17B10 (0.61) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL21275460 0.88 RAB9A (0.76) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL9281809 0.87 GFER (0.76) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
Naptalam SCHEMBL8382453 0.87 HSD17B10 (0.58) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL4926868 0.85 KDM4E (0.72) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL12172779 0.85 GFER (0.69) HSD17B10CHRNB2CHRNB4CHRNA3CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 12760 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12568967-B2 Compositions comprising pyridine carboxylate herbicides with synthetic auxin herbicides or auxin transport inhibitors CORTEVA AGRISCIENCE LLC (US) 2026-03-10 US claimed
US-20260007133-A1 HERBICIDAL COMPOSITION COMPRISING AZINE COMPOUNDS BASF SE (DE) 2026-01-08 US claimed
US-20250374920-A1 HERBICIDAL COMPOSITION COMPRISING ALKYL POLYGLYCOSIDES BASF SE (DE) 2025-12-11 US claimed
US-20250366479-A1 Non-Aqueous Organo Liquid Delivery Systems containing dispersed Organo Polycarboxylate Functionalities that improves efficiencies and properties of nitrogen sources SOILGENIC TECH LLC (US) 2025-12-04 US claimed
EP-3060043-B1 PESTICIDAL COMPOSITIONS AND RELATED METHODS CORTEVA AGRISCIENCE LLC (US) 2025-11-26 EP claimed
EP-3578542-B1 COMPOSITIONS HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-11-12 EP claimed
EP-4646109-A2 NATURAL LIPID PARTICLE FORMULATIONS FOR AGRICULTURAL APPLICATIONS Invaio Sciences, Inc. (US) 2025-11-12 EP claimed
US-20250318528-A1 HERBICIDE COMPOSITION AND WEED CONTROLLING METHOD SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2025-10-16 US claimed
EP-3578543-B1 COMPOSITIONS COMPRISING MOLECULES HAVING PESTICIDAL UTILITY AND PROCESSES RELATED THERETO CORTEVA AGRISCIENCE LLC (US) 2025-08-20 EP claimed
US-12391729-B2 Fusion proteins, recombinant bacteria, and methods for using recombinant bacteria SPOGEN BIOTECH INC. (US) 2025-08-19 US claimed
EP-0063866-B1 QUINOLIN-3-YLOXY(AMINO)PHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, PROCESS FOR THEIR SYNTHESIS, HERBICIDAL COMPOSITIONS CONTAINING THEM, AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1987-12-09 EP claimed
EP-0238240-A2 Dry reactive processing UNIROYAL CHEMICAL COMPANY, Inc. (US) 1987-09-23 EP claimed
EP-0212200-A2 Pyridine derivatives and herbicidal composition NISSAN CHEMICAL INDUSTRIES LTD. (JP) 1987-03-04 EP claimed
CN-86105501-A Pyridine derivate and preparation method thereof and herbicidal composition 1987-01-21 CN claimed
EP-0207653-A1 Herbicidal compositions comprising microbial herbicides and chemical herbicides or plant growth regulators THE UNIVERSITY OF VERMONT AND STATE AGRICULTURAL COLLEGE (US) 1987-01-07 EP claimed
EP-0029319-B1 QUINOLINYLOXY(AMINO)PHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, PROCESS FOR THEIR SYNTHESIS, HERBICIDAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1986-01-15 EP claimed
EP-0060607-B1 2-(2-HALO-4-(6-HALOQUINOXALIN-2-YLOXY)PHENOXY)PROPIONATES, PROCESS FOR THEIR SYNTHESIS, HERBICIDAL COMPOSITIONS CONTAINING THEM AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1985-08-28 EP claimed
EP-0004414-B1 MIXTURES OF HERBICIDAL PYRIDYLOXYPHENOXYPROPANOIC ACID DERIVATIVES WITH OTHER HERBICIDES, AND PROCESSES OF KILLING UNWANTED PLANTS THEREWITH IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-07-24 EP claimed
EP-0023785-B1 QUINOXALINYLOXYPHENOXYALKANE CARBOXYLIC ACID DERIVATIVES, THEIR PREPARATION AND THEIR USE AS HERBICIDES ICI AUSTRALIA LIMITED (AU) 1985-04-03 EP claimed
EP-0004414-A1 Mixtures of herbicidal pyridyloxyphenoxypropanoic acid derivatives with other herbicides, and processes of killing unwanted plants therewith IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1979-10-03 EP claimed