SCHEMBL5495317

SCHEMBL5495317

O=C(O)C1(NS(=O)(=O)c2cccs2)C[C@H]1c1ccccc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADAMTS5 Q9UNA0 6/20 0.59
CYP2C19 P33261 2/20 0.49
MAPK1 P28482 1/20 0.49
SLC1A3 P43003 1/20 0.43
SLC1A2 P43004 1/20 0.43
SLC1A1 P43005 1/20 0.43
TSHR P16473 1/20 0.41
ALDH1A1 P00352 2/20 0.41
GAA P10253 1/20 0.41
TP53 P04637 1/20 0.41
HSD11B1 P28845 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
PSEN1 P49768 1/20 0.40
PSEN2 P49810 1/20 0.40
APH1B Q8WW43 1/20 0.40
NCSTN Q92542 1/20 0.40
APH1A Q96BI3 1/20 0.40
PSENEN Q9NZ42 1/20 0.40
BRAF P15056 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2765348 1.00 ADAMTS5 (0.59) ADAMTS5CYP2C19MAPK1SLC1A3SLC1A2
SCHEMBL2765349 1.00 ADAMTS5 (0.59) ADAMTS5CYP2C19MAPK1SLC1A3SLC1A2
SCHEMBL2765675 0.81 ADAMTS5 (0.69) ADAMTS5CYP2C19MAPK1ALDH1A1
SCHEMBL2765671 0.81 ADAMTS5 (0.69) ADAMTS5CYP2C19MAPK1ALDH1A1
SCHEMBL5494344 0.81 ADAMTS5 (0.69) ADAMTS5CYP2C19MAPK1ALDH1A1
SCHEMBL5492303 0.80 ADAMTS5 (0.66) ADAMTS5CYP2C19MAPK1
SCHEMBL2763926 0.80 ADAMTS5 (0.66) ADAMTS5CYP2C19MAPK1ALDH1A1MEN1
SCHEMBL2763988 0.80 ADAMTS5 (0.66) ADAMTS5CYP2C19MAPK1
SCHEMBL2765101 0.80 ADAMTS5 (0.66) ADAMTS5CYP2C19MAPK1ALDH1A1MEN1
SCHEMBL2763922 0.80 ADAMTS5 (0.66) ADAMTS5CYP2C19MAPK1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007516982-A 2007-06-28 JP claimed
EP-1694410-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF Japan Tobacco, Inc. (JP) 2006-08-30 EP claimed
WO-2005058884-A2 CYCLOPROPANE COMPOUNDS AND PHARMACEUTICAL USE THEREOF JAPAN TOBACCO INC. (JP) 2005-06-30 WO claimed