SCHEMBL5497003

SCHEMBL5497003

CC(Oc1ccc(SCC#Cc2ccccc2C(F)(F)F)cc1)C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 8/20 0.43
PPARD Q03181 1/20 0.43
CYP1A2 P05177 1/20 0.43
GAA P10253 1/20 0.43
CYP2C9 P11712 1/20 0.43
PKM P14618 1/20 0.43
CYP2C19 P33261 1/20 0.43
PPARG P37231 8/20 0.39
PDK2 Q15119 1/20 0.39
FFAR1 O14842 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.37
ADRB3 P13945 5/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5497621 0.74 EPHX2 (0.46) PPARAPPARDCYP1A2GAACYP2C9
SCHEMBL5486731 0.73 PTGDR2 (0.57) PPARAPPARDPPARGPTGDR2
SCHEMBL5490364 0.72 PTGDR2 (0.56) PPARAPPARDPPARGPTGDR2
SCHEMBL11151598 0.70 CYP1A2 (0.55) PPARACYP1A2GAACYP2C9PKM
SCHEMBL5496562 0.70 PPARD (0.52) PPARAPPARDCYP1A2GAACYP2C9
SCHEMBL5488425 0.68 PTGDR2 (0.44) PPARAPPARDPPARGPTGDR2
SCHEMBL10944856 0.68 PPARA (0.56) PPARAPPARDCYP1A2GAACYP2C9
SCHEMBL9780575 0.67 PPARG (0.60) PPARACYP1A2GAACYP2C9PKM
SCHEMBL9780582 0.67 PPARG (0.60) PPARACYP1A2GAACYP2C9PKM
SCHEMBL25212758 0.66 CYP1A2 (0.59) PPARAPPARDCYP1A2GAACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765760-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F.HOFFMANN-LA ROCHE AG (CH) 2007-03-28 EP claimed
WO-2006002802-A1 PHENYL DERIVATIVES COMPRISING AN ACETYLENE GROUP F. HOFFMANN-LA ROCHE AG (CH) 2006-01-12 WO claimed