SCHEMBL5497325

SCHEMBL5497325

CCOCCc1c[nH]c2cc(NNc3ccc4c(CCOCC)c[nH]c4c3)ccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 6/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA7 P36544 1/20 0.43
CHRNA4 P43681 1/20 0.43
NPC1 O15118 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
HTR1A P08908 2/20 0.41
HTR6 P50406 2/20 0.41
HTR2C P28335 3/20 0.40
HTR2B P41595 2/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
SPR P35270 1/20 0.39
CFTR P13569 1/20 0.39
SLC6A4 P31645 1/20 0.38
HTR3E A5X5Y0 1/20 0.38
HTR3B O95264 1/20 0.38
HTR1D P28221 1/20 0.38
HTR1B P28222 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15074675 0.82 HTR2A (0.63) HTR2ACHRNB2CHRNA7CHRNA4NPC1
SCHEMBL397322 0.81 HTR2A (0.50) HTR2ACHRNB2CHRNA7CHRNA4MEN1
SCHEMBL5497322 0.81 HTR2A (0.50) HTR2ACHRNB2CHRNA7CHRNA4MEN1
SCHEMBL11924512 0.81 HTR1A (0.51) HTR2ACHRNB2CHRNA7CHRNA4NPC1
SCHEMBL5484718 0.80 CFTR (0.53) HTR2ACHRNB2CHRNA7CHRNA4NPC1
SCHEMBL8957544 0.79 HTR1D (0.51) HTR2ACHRNB2CHRNA7CHRNA4NPC1
SCHEMBL13651810 0.77 HTR2A (0.58) HTR2AMEN1KMT2AHTR1AHTR6
SCHEMBL9001726 0.77 HTR1D (0.40) HTR2ACHRNB2CHRNA7CHRNA4NPC1
SCHEMBL398456 0.75 CFTR (0.78) CFTR
SCHEMBL25082440 0.71 HTR2A (0.68) HTR2AHTR1AHTR6HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed