SCHEMBL5497322

SCHEMBL5497322

CCOCCc1c[nH]c2cc(N)ccc12.CCOCCc1c[nH]c2cc(N)ccc12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 7/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
HTR2C P28335 4/20 0.47
HTR1A P08908 8/20 0.43
HTR1B P28222 8/20 0.43
CYP2C19 P33261 2/20 0.43
HPGD P15428 1/20 0.43
HTR6 P50406 3/20 0.42
HTR1D P28221 7/20 0.41
CYP1A2 P05177 3/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2D6 P10635 2/20 0.41
NFKB1 P19838 2/20 0.41
HTR7 P34969 2/20 0.41
MPO P05164 1/20 0.41
CYP2A6 P11509 1/20 0.41
CTSK P43235 1/20 0.41
CYP2A13 Q16696 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL397322 1.00 HTR2A (0.50) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL15074675 0.84 HTR2A (0.63) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL11924512 0.82 HTR1A (0.51) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL5497325 0.81 HTR2A (0.43) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL5145582 0.80 HTR2A (0.54) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL8957544 0.80 HTR1D (0.51) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL398434 0.79 HTR2A (0.51) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL5484715 0.79 HTR2A (0.51) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL27797581 0.79 HPGD (0.49) HTR2AMEN1KMT2AHTR2CHTR1A
SCHEMBL13651810 0.78 HTR2A (0.58) HTR2AMEN1KMT2AHTR2CHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773816-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmaceuticals Incorporated (US) 2007-04-18 EP disclosed
WO-2006002421-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2006-01-05 WO disclosed