SCHEMBL5498052

SCHEMBL5498052

COc1ccc(C(=O)OCC2CC2)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
MAPT P10636 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
ALDH1A1 P00352 1/20 0.53
ESR2 Q92731 1/20 0.53
NPC1 O15118 3/20 0.50
RAB9A P51151 3/20 0.50
PARP15 Q460N3 1/20 0.49
PARP10 Q53GL7 1/20 0.49
PARP2 Q9UGN5 1/20 0.49
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
PTGIR P43119 1/20 0.48
PTGDR Q13258 1/20 0.48
ADRB2 P07550 1/20 0.48
ADRB1 P08588 1/20 0.48
ADRB3 P13945 1/20 0.48
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13498610 1.00 CA1 (0.55) CA1CA2MAPTSMN1; SMN2ALDH1A1
SCHEMBL18461191 0.94 SMN1; SMN2 (0.54) CA1CA2MAPTSMN1; SMN2ALDH1A1
SCHEMBL19214417 0.90 ALDH1A1 (0.51) CA1CA2MAPTSMN1; SMN2ALDH1A1
SCHEMBL12561798 0.88 CARM1 (0.52) CA1CA2MAPTSMN1; SMN2ALDH1A1
SCHEMBL17204382 0.84 CA1 (0.51) CA1CA2MAPTSMN1; SMN2ALDH1A1
SCHEMBL23928027 0.83 CARM1 (0.48) CA1CA2MAPTESR2RAB9A
SCHEMBL13498612 0.83 RAB9A (0.50) CA1CA2MAPTALDH1A1ESR2
SCHEMBL14665431 0.83 CARM1 (0.48) CA1CA2ESR2RAB9APARP15
SCHEMBL11843612 0.83 RAB9A (0.50) CA1CA2MAPTALDH1A1ESR2
SCHEMBL19407121 0.83 MAPT (0.63) MAPTSMN1; SMN2ALDH1A1ESR2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1740545-A1 PROCESS FOR MAKING MONTELUKAST AND INTERMEDIATES THEREFOR Synthon B.V. (NL) 2007-01-10 EP disclosed
WO-2005105750-A1 PROCESS FOR MAKING MONTELUKAST AND INTERMEDIATES THEREFOR SYNTHON B.V. (NL) 2005-11-10 WO disclosed
US-3975429-A Cyclopropanemethyl esters of cinnamic acid and derivatives thereof ZOECON CORPORATION (US) 1976-08-17 US disclosed