SCHEMBL5499100

SCHEMBL5499100

OC1(CCCc2cccc(F)c2C(F)(F)F)CCNCC1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 7/20 0.41
SLC6A4 P31645 3/20 0.41
SLC6A2 P23975 2/20 0.41
CYP2D6 P10635 1/20 0.41
TACR1 P25103 2/20 0.37
HTR2C P28335 1/20 0.33
P2RX7 Q99572 1/20 0.33
REN P00797 5/20 0.32
CYP3A4 P08684 5/20 0.32
GPR4 P46093 1/20 0.31
CMA1 P23946 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4390004 0.84 FFAR4 (0.39) KCNH2SLC6A4SLC6A2TACR1HTR2C
SCHEMBL2785289 0.82 FFAR4 (0.43) SLC6A4SLC6A2TACR1HTR2CP2RX7
SCHEMBL5499318 0.82 KCNH2 (0.33) KCNH2SLC6A4SLC6A2CYP2D6TACR1
SCHEMBL5500092 0.79 FFAR4 (0.43) KCNH2SLC6A4SLC6A2TACR1P2RX7
SCHEMBL5502120 0.77 SLC6A2 (0.38) KCNH2SLC6A4SLC6A2CYP2D6TACR1
SCHEMBL5493818 0.76 FFAR4 (0.41) KCNH2SLC6A4SLC6A2TACR1HTR2C
SCHEMBL5495876 0.75 FFAR4 (0.38) SLC6A4SLC6A2HTR2CREN
SCHEMBL27618109 0.75 TAAR1 (0.43) SLC6A4SLC6A2CYP2D6HTR2CCYP3A4
SCHEMBL5499363 0.74 TACR1 (0.43) SLC6A4SLC6A2TACR1HTR2CP2RX7
Hydrochloric Acid SCHEMBL1475155 0.74 TAAR1 (0.42) SLC6A4SLC6A2CYP2D6HTR2CCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1773772-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-04-18 EP disclosed
WO-2005121087-A1 NEW DISUBSTITUTED PHENYLPIPERIDINES/PIPERAZINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO disclosed