SCHEMBL5502870

SCHEMBL5502870

[CH2]C(CCCc1ccccc1)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 3/20 0.50
SIGMAR1 Q99720 4/20 0.44
MAOA P21397 1/20 0.43
CHRM2 P08172 1/20 0.42
HTR1A P08908 1/20 0.42
ADRA2A P08913 1/20 0.42
CHRM1 P11229 1/20 0.42
DRD1 P21728 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
ADRA1A P35348 1/20 0.42
OPRM1 P35372 1/20 0.42
DRD3 P35462 1/20 0.42
SLC6A3 Q01959 1/20 0.42
CNR1 P21554 1/20 0.42
MAOB P27338 1/20 0.42
HTR2A P28223 1/20 0.42
ACP3 P15309 1/20 0.42
GRIK1 P39086 1/20 0.41
IDO1 P14902 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11300940 0.92 KCNH2 (0.47) KCNH2SIGMAR1MAOAMAOBHTR2A
SCHEMBL1147908 0.87 ACP3 (0.48) KCNH2SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL11365631 0.84 HDAC1 (0.48) KCNH2SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL4952239 0.81 FDFT1 (0.50)
SCHEMBL9132974 0.80 KCNH2 (0.66) KCNH2SIGMAR1MAOACHRM2HTR1A
SCHEMBL11305200 0.79 HDAC1 (0.44) KCNH2SIGMAR1SLC6A2SLC6A4SLC6A3
SCHEMBL7374792 0.79 SIGMAR1 (0.49) SIGMAR1MAOB
SCHEMBL10655335 0.79 KCNH2 (0.46) KCNH2SIGMAR1MAOACHRM2HTR1A
SCHEMBL3020787 0.78 HRH1 (0.40) KCNH2SIGMAR1HTR2A
SCHEMBL4951030 0.77 ACP3 (0.41) KCNH2SIGMAR1SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1848692-A1 AZOLYLACYLGUANIDINES AS ß-SECRETASE INHIBITORS Wyeth (US) 2007-10-31 EP disclosed
WO-2006088711-A1 AZOLYLACYLGUANIDINES AS β-SECRETASE INHIBITORS WYETH (US) 2006-08-24 WO disclosed
US-5110865-A Fiber treatment, lubricants, release agents, antifoam agents, lustrants TORAY SILICONE COMPANY, LTD. (JP) 1992-05-05 US disclosed