SCHEMBL5503113

SCHEMBL5503113

O=C(O)C(Cc1cscn1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 7/20 0.52
SLC6A2 P23975 2/20 0.46
SLC6A4 P31645 1/20 0.46
GPR142 Q7Z601 4/20 0.45
POLB P06746 1/20 0.43
CAPN1 P07384 1/20 0.43
CYP2C19 P33261 1/20 0.42
P4HTM Q9NXG6 1/20 0.41
CTSB P07858 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
EPHX1 P07099 1/20 0.39
OPRD1 P41143 1/20 0.39
KDM4C Q9H3R0 1/20 0.38
FOLH1 Q04609 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9565308 0.78 KDM4E (0.44) SLC6A3SLC6A2SLC6A4GPR142CAPN1
SCHEMBL7280731 0.77 CYP1A2 (0.61) SLC6A3GPR142FOLH1
SCHEMBL7829956 0.76 PTPRA (0.65) SLC6A4POLBCYP2C19P4HTMEPHX1
SCHEMBL7829954 0.76 PTPRA (0.65) SLC6A4POLBCYP2C19P4HTMEPHX1
SCHEMBL14561302 0.73 GPR142 (0.40) SLC6A3GPR142CAPN1CTSBCTSS
SCHEMBL22193474 0.73 GPR142 (0.40) SLC6A3SLC6A2SLC6A4GPR142CAPN1
SCHEMBL6897379 0.73 GPR142 (0.40) SLC6A3SLC6A2SLC6A4GPR142CAPN1
SCHEMBL990477 0.73 DPP4 (0.49) SLC6A3GPR142POLBOPRD1
SCHEMBL6897376 0.73 GPR142 (0.40) SLC6A3SLC6A2SLC6A4GPR142CAPN1
SCHEMBL5535517 0.73 GPR142 (0.40) SLC6A3GPR142CAPN1CTSBCTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1786792-A2 THIAZOLE DERIVATIVES HAVING VAP-1 INHIBITORY ACTIVITY Astellas Pharma Inc. (JP) 2007-05-23 EP disclosed
WO-2006011631-A2 THIAZOLE DERIVATIVES HAVING VAP-1 INHIBITORY ACTIVITY ASTELLAS PHARMA INC. (JP) 2006-02-02 WO disclosed