SCHEMBL5503573

SCHEMBL5503573

CNc1nc(N)c2ccc(-c3ccccc3C(F)(F)F)cc2n1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 1/20 0.51
DHFR P00374 4/20 0.48
TRPA1 O75762 3/20 0.46
PTPN1 P18031 2/20 0.46
CYP1A2 P05177 6/20 0.44
CYP2C19 P33261 5/20 0.44
CYP2D6 P10635 4/20 0.44
RECQL P46063 1/20 0.44
SCN5A Q14524 1/20 0.44
SCN9A Q15858 1/20 0.44
CYP3A4 P08684 5/20 0.44
USP2 O75604 3/20 0.44
TSHR P16473 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPK1 P28482 2/20 0.44
CLK4 Q9HAZ1 2/20 0.44
PIK3R1 P27986 1/20 0.44
PIK3CA P42336 1/20 0.44
ALOX5AP P20292 1/20 0.44
FEN1 P39748 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4532433 0.84 DHFR (0.68) BACE1DHFRTRPA1SCN5ASCN9A
SCHEMBL4528905 0.81 PTPN1 (0.62) BACE1DHFRTRPA1PTPN1CYP1A2
SCHEMBL4524134 0.74 CYP1A2 (0.57) BACE1DHFRTRPA1PTPN1CYP1A2
SCHEMBL14529155 0.72 CYP1A2 (0.49) BACE1CYP1A2CYP2C19CYP2D6RECQL
SCHEMBL6978694 0.71 NPC1 (0.64) TSHRALDH1A1MAPK1MEN1KMT2A
SCHEMBL4528846 0.70 PTPN1 (0.66) BACE1DHFRPTPN1CYP1A2CYP2C19
SCHEMBL12907209 0.69 SCN5A (0.59) BACE1TRPA1SCN5ASCN9ACYP3A4
SCHEMBL3735069 0.69 BACE1 (0.60) BACE1TRPA1CYP1A2CYP2C19CYP2D6
Trifluoroacetic Acid SCHEMBL4527702 0.69 CYP2D6 (0.51) BACE1DHFRTRPA1PTPN1CYP1A2
SCHEMBL28403515 0.68 AR (0.56) BACE1TRPA1CYP1A2CYP2C19CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812409-A1 AMINOQUINAZOLINES COMPOUNDS F. Hoffmann-Roche AG (CH) 2007-08-01 EP claimed
WO-2006050843-A1 AMINOQUINAZOLINES COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-18 WO claimed
EP-1812409-A1 AMINOQUINAZOLINES COMPOUNDS F. Hoffmann-Roche AG (CH) 2007-08-01 EP disclosed
WO-2006050843-A1 AMINOQUINAZOLINES COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-18 WO disclosed