SCHEMBL5504510

SCHEMBL5504510

O=C(O)c1cc(OCCCC2CNCCN2c2cccc3sccc23)c2ccccc2n1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 5/20 0.38
DRD2 P14416 5/20 0.38
HTR2A P28223 5/20 0.38
ALOX15 P16050 1/20 0.37
HTR2C P28335 2/20 0.36
ADRA1A P35348 2/20 0.36
HRH1 P35367 2/20 0.36
ADRB2 P07550 1/20 0.34
ADRB1 P08588 1/20 0.34
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
DRD1 P21728 1/20 0.34
DRD4 P21917 1/20 0.34
DRD5 P21918 1/20 0.34
SLC6A2 P23975 1/20 0.34
ADRA1D P25100 1/20 0.34
HTR1D P28221 1/20 0.34
HTR1B P28222 1/20 0.34
HTR1E P28566 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511426 0.94 HTR1A (0.37) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL1037492 0.78 HTR1A (0.57) HTR1ADRD2HTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL1037712 0.77 HTR1A (0.56) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL4630514 0.76 DRD2 (0.33) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL5506910 0.73 MAP2K1 (0.44) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL5508733 0.73 DRD2 (0.45) HTR1ADRD2HTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL4630605 0.73 HTR1A (0.33) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL5502282 0.72 DRD2 (0.43) HTR1ADRD2HTR2AHTR2CADRA1A
SCHEMBL20915099 0.72 DRD2 (0.46) HTR1ADRD2HTR2AHTR2CADRA1A
Hydrochloric Acid SCHEMBL5512177 0.72 DRD2 (0.42) HTR1ADRD2HTR2AHTR2CADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869025-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENES FOR TREATMENT OF MENTAL DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-12-26 EP disclosed
WO-2006112464-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENES FOR TREATMENT OF MENTAL DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-10-26 WO disclosed