SCHEMBL5504528

SCHEMBL5504528

CCN(CC)S(=O)(=O)n1cc(-c2ccc3ccccc3c2)nc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.41
LMNA P02545 2/20 0.41
CTRC Q99895 1/20 0.40
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
CA1 P00915 2/20 0.38
CA2 P00918 2/20 0.38
CA9 Q16790 2/20 0.38
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38
TUBA1C Q9BQE3 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3747955 0.85 SMN1; SMN2 (0.43) KDM4ELMNACTRCRAB9ANPC1
SCHEMBL4728696 0.66 KDM4E (0.48) KDM4ELMNARAB9ANPC1ALDH1A1
SCHEMBL11978725 0.65 CTRC (0.61) KDM4ELMNACTRCRAB9ANPC1
SCHEMBL5504526 0.65 BACE1 (0.43) CYP1A2
SCHEMBL3747965 0.64 CYP2C9 (0.51) KDM4ECTRCRAB9ANPC1TUBB4A
SCHEMBL20021989 0.64 CNR2 (0.62) LMNARAB9ANPC1ALDH1A1RXFP1
SCHEMBL13831046 0.62 CYP1A2 (0.46) KDM4ELMNACTRCRAB9ANPC1
SCHEMBL19656044 0.62 KMT2A (0.46) KDM4ERAB9ANPC1CA1CA2
SCHEMBL1691846 0.62 NPC1 (0.68) KDM4ELMNARAB9ANPC1ALDH1A1
SCHEMBL16805046 0.62 CYP1A2 (0.63) KDM4ECTRCRAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1791833-A2 4-(CONDENSED CYCLICMETHYL)-IMIDAZOLE-2-THIONES ACTING AS ALPHA2 ADRENERGIC AGONISTS Allergan, Inc. (US) 2007-06-06 EP disclosed
WO-2006036497-A2 4-(CONDENSED CYCLICMETHYL)-IMIDAZOLE-2-THIONES ACTING AS ALPHA2 ADRENERGIC AGONISTS ALLERGAN, INC. (US) 2006-04-06 WO disclosed