SCHEMBL5505202

SCHEMBL5505202

CC1CCCN(CCCN2[C]N(CCCN3CCCC3C)CC2)C1

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 14/20 0.39
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
MAOB P27338 2/20 0.37
HRH2 P25021 1/20 0.37
HRH1 P35367 1/20 0.37
HTR7 P34969 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502805 0.96 HRH3 (0.36) HRH3CHRM2CHRM1KDM4E
SCHEMBL5502044 0.89 HRH3 (0.35) HRH3
SCHEMBL5507033 0.88 HRH3 (0.42) HRH3
SCHEMBL5508033 0.87 HRH3 (0.42) HRH3
SCHEMBL5502491 0.85 CXCR4 (0.39) HRH3CHRM2CHRM1MAOBHRH2
SCHEMBL5501715 0.85 HRH3 (0.34) HRH3
SCHEMBL5508184 0.84 HRH3 (0.41) HRH3CHRM2CHRM1MAOBHRH2
SCHEMBL5505204 0.84 HRH3 (0.41) HRH3MAOBHRH2HRH1HTR7
SCHEMBL5502174 0.84 HRH3 (0.44) HRH3
SCHEMBL5504695 0.84 HRH3 (0.40) HRH3CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847530-A1 DIAMINE DERIVATIVE KYOWA HAKKO KOGYO CO., LTD. (JP) 2007-10-24 EP disclosed