SCHEMBL5505220

SCHEMBL5505220

O=C(O)[C@H](CS)NCc1ccc(-c2ccccc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MME P08473 8/20 0.49
ACE P12821 7/20 0.49
ACE2 Q9BYF1 7/20 0.49
CPA1 P15085 5/20 0.49
LMNA P02545 3/20 0.49
ALDH1A1 P00352 2/20 0.49
HTT P42858 2/20 0.48
MAPK1 P28482 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
SRR Q9GZT4 2/20 0.47
PSAT1 Q9Y617 2/20 0.47
EPHX2 P34913 1/20 0.46
NR1H4 Q96RI1 1/20 0.46
FFAR1 O14842 1/20 0.46
ABCC4 O15439 1/20 0.46
GAA P10253 1/20 0.46
TSHR P16473 1/20 0.46
PTGS1 P23219 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1109641 0.91 CPA3 (0.50) MMEGAA
SCHEMBL1031027 0.91 CPA3 (0.50) MMEGAA
SCHEMBL515921 0.91 CPA3 (0.50) MMEGAA
Hydrochloric Acid SCHEMBL28182328 0.90 CPA3 (0.49) MMEGAA
Hydrochloric Acid SCHEMBL1927540 0.90 CPA3 (0.49) MMEGAA
Hydrochloric Acid SCHEMBL1927541 0.90 CPA3 (0.49) MMEGAA
Benzenemethanethiol SCHEMBL11584239 0.87 IDO1 (0.47) MMEGAA
SCHEMBL7614779 0.83 ACE (0.49) ACELMNAFFAR1
SCHEMBL2328314 0.83 ACE (0.49) ACELMNAFFAR1
SCHEMBL1760830 0.83 ALDH1A1 (0.50) MMEACELMNAALDH1A1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833978-A1 TRIPEPTIDE AND TETRAPEPTIDE THIOETHERS TELIK, INC. (US) 2007-09-19 EP disclosed
WO-2006074249-A1 TRIPEPTIDE AND TETRAPEPTIDE THIOETHERS TELIK, INC. (US) 2006-07-13 WO disclosed