SCHEMBL5506579

SCHEMBL5506579

CCOC(=O)c1cc(S(=O)(=O)N2CCCC2)c(C)cc1OCC.CCOC(=O)c1cc(S(=O)(=O)N2CCCCC2)c(C)cc1OCC.CCOc1cc(OC)c(S(=O)(=O)N2CCCCC2)cc1C(=O)O

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.58
TDP1 Q9NUW8 1/20 0.54
KMT2A Q03164 6/20 0.52
ALDH1A1 P00352 6/20 0.52
MEN1 O00255 4/20 0.52
TSHR P16473 7/20 0.51
GAA P10253 1/20 0.51
NPBWR1 P48145 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.51
POLB P06746 2/20 0.49
HTT P42858 1/20 0.45
MCOLN3 Q8TDD5 1/20 0.45
MAPK1 P28482 1/20 0.44
HSD17B10 Q99714 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4004183 0.92 TSHR (0.60) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL3998128 0.90 KDM4E (0.71) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL4001104 0.89 KDM4E (0.69) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL1546461 0.83 TSHR (0.59) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL11184423 0.83 KMT2A (0.68) KDM4EKMT2AALDH1A1MEN1TSHR
SCHEMBL11178802 0.81 KMT2A (0.65) KDM4EKMT2AALDH1A1MEN1TSHR
SCHEMBL11180002 0.81 TSHR (0.73) KDM4EKMT2AALDH1A1MEN1TSHR
SCHEMBL4006356 0.80 ALDH1A1 (0.61) KDM4ETDP1KMT2AALDH1A1MEN1
SCHEMBL3997775 0.79 ALDH1A1 (0.64) KDM4ETDP1KMT2AALDH1A1TSHR
SCHEMBL3999221 0.79 ALDH1A1 (0.62) KDM4ETDP1KMT2AALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861376-A1 CIS-2,4,5-TRIARYL-IMIDAZOLINES AND THEIR USE AS ANTI-CANCER MEDICAMENTS F. Hoffmann-Roche AG (CH) 2007-12-05 EP disclosed
WO-2006097261-A1 CIS-2,4,5-TRIARYL-IMIDAZOLINES AND THEIR USE AS ANTI-CANCER MEDICAMENTS F.HOFFMANN-LA ROCHE AG (CH) 2006-09-21 WO disclosed