SCHEMBL5506770

SCHEMBL5506770

Cc1nc2c3c(c(C(=S)N(C)C)cc2[nH]1)CC[C@@H](c1ccccc1)O3

nearest known ligand 0.34

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 7/20 0.34
ATP4A P20648 1/20 0.32
ATP4B P51164 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5106333 0.88 DHODH (0.39) DHODH
SCHEMBL4664674 0.88 DHODH (0.39) DHODH
Oxalic Acid SCHEMBL5657472 0.87 DHODH (0.38) DHODH
SCHEMBL5511902 0.80 ATP4A (0.33) ATP4AATP4B
SCHEMBL5507104 0.80 ATP4A (0.33) ATP4AATP4B
SCHEMBL1943187 0.79 DHODH (0.33) DHODH
SCHEMBL4961983 0.77 DHODH (0.35) DHODH
SCHEMBL5507799 0.76 PARP1 (0.32) ATP4AATP4B
SCHEMBL5425360 0.72 ATP4A (0.43) ATP4AATP4B
SCHEMBL5506546 0.69 ATP4A (0.35) ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863820-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES Nycomed GmbH (DE) 2007-12-12 EP claimed
WO-2006100255-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES NYCOMED GMBH (DE) 2006-09-28 WO claimed
EP-1863820-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES Nycomed GmbH (DE) 2007-12-12 EP disclosed
WO-2006100255-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES NYCOMED GMBH (DE) 2006-09-28 WO disclosed