SCHEMBL5507799

SCHEMBL5507799

CN(C)C(=S)c1cc2c(nc(C3CC3)n2C)c2c1CCC(c1ccccc1)O2

nearest known ligand 0.32

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.32
TLR7 Q9NYK1 1/20 0.31
BRD4 O60885 1/20 0.31
ATP4A P20648 1/20 0.31
ATP4B P51164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4664631 0.89 PARP1 (0.36) PARP1TLR7BRD4ATP4AATP4B
SCHEMBL5507104 0.89 ATP4A (0.33) ATP4AATP4B
SCHEMBL5511902 0.89 ATP4A (0.33) ATP4AATP4B
Dimethylamine SCHEMBL5505793 0.81
SCHEMBL5506546 0.79 ATP4A (0.35) ATP4AATP4B
SCHEMBL4664616 0.77 RIPK1 (0.36) BRD4ATP4AATP4B
SCHEMBL4662902 0.77 RIPK1 (0.36) BRD4ATP4AATP4B
SCHEMBL4663156 0.77 RIPK1 (0.36) BRD4ATP4AATP4B
SCHEMBL5506770 0.76 DHODH (0.34) ATP4AATP4B
SCHEMBL5511615 0.76 ATP4A (0.33) ATP4AATP4B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863820-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES Nycomed GmbH (DE) 2007-12-12 EP disclosed
WO-2006100255-A1 THIOAMIDE-SUBSTITUTED TRICYCLIC BENZIMIDAZOLES USEFUL FOR THE TREATMENT OF GASTROINTESTINAL DISEASES NYCOMED GMBH (DE) 2006-09-28 WO disclosed