SCHEMBL5509065

SCHEMBL5509065

C#C[C@H]1O[C@H](n2cnc3c(NC4CCCC4)ncnc32)[C@@H]2OC(C)(C)O[C@@H]21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.52
ADORA3 P0DMS8 3/20 0.52
ADORA2A P29274 3/20 0.52
PMP22 Q01453 2/20 0.52
ADORA2B P29275 2/20 0.52
ADORA1 P30542 2/20 0.52
GAA P10253 1/20 0.52
HTT P42858 1/20 0.52
SIGMAR1 Q99720 1/20 0.52
SLC29A1 Q99808 1/20 0.52
RXFP1 Q9HBX9 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
TP53 P04637 1/20 0.52
NFKB1 P19838 1/20 0.52
HIF1A Q16665 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 1/20 0.51
CYP2C19 P33261 1/20 0.51
THPO P40225 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5504161 1.00 TSHR (0.52) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5504164 1.00 TSHR (0.52) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5509240 1.00 TSHR (0.52) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5513305 0.99 ADORA2A (0.52) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5513298 0.99 ADORA2A (0.52) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5509613 0.98 ADORA3 (0.49) TSHRADORA3ADORA2APMP22ADORA2B
SCHEMBL5503453 0.91 ADORA1 (0.49) ADORA3ADORA2AADORA2BADORA1SLC29A1
SCHEMBL5503445 0.91 ADORA1 (0.49) ADORA3ADORA2AADORA2BADORA1SLC29A1
SCHEMBL5505648 0.89 ADORA1 (0.54) ADORA3ADORA2AADORA2BADORA1SLC29A1
SCHEMBL5505653 0.89 ADORA1 (0.54) ADORA3ADORA2AADORA2BADORA1SLC29A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537133-B1 PARTIAL AND FULL AGONISTS OF A1 ADENOSINE RECEPTORS CV THERAPEUTICS INC (US) 2007-07-25 EP disclosed