SCHEMBL5509255

SCHEMBL5509255

CS(=O)(=O)Nc1cc(Cl)c(CNC(=O)O)cc1I

nearest known ligand 0.44

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.44
RCE1 Q9Y256 1/20 0.44
EPHX2 P34913 14/20 0.40
NR1H4 Q96RI1 12/20 0.40
PPARG P37231 1/20 0.40
TRPV1 Q8NER1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2001184 0.83 EPHX2 (0.41) ALDH1A1KDM4ERCE1EPHX2NR1H4
SCHEMBL2002663 0.83 EPHX2 (0.43) ALDH1A1KDM4ERCE1EPHX2NR1H4
SCHEMBL5509325 0.81 ALDH1A1 (0.42) ALDH1A1KDM4ERCE1EPHX2NR1H4
SCHEMBL2003851 0.79 PIK3CD (0.39) ALDH1A1KDM4ERCE1EPHX2NR1H4
SCHEMBL2002176 0.78 EPHX2 (0.52) EPHX2NR1H4PPARG
SCHEMBL2952173 0.75 KDM4E (0.47) ALDH1A1KDM4E
SCHEMBL28772365 0.74 SMN1; SMN2 (0.41) ALDH1A1KDM4ERCE1EPHX2NR1H4
SCHEMBL15608399 0.74 EPHX2 (0.38) ALDH1A1KDM4EEPHX2NR1H4
SCHEMBL5502890 0.73 EPHX2 (0.35) EPHX2NR1H4
SCHEMBL980032 0.70 PIK3CD (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861358-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2007-12-05 EP disclosed
WO-2006101321-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2006-09-28 WO disclosed