SCHEMBL5509732

SCHEMBL5509732

COCCCN1C(=O)COc2ccc(COC3CN[C@H](CO)CC3c3ccc(OC)cc3)cc21

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
REN P00797 4/20 0.42
MAPT P10636 2/20 0.41
CYP3A4 P08684 2/20 0.40
SMPD1 P17405 1/20 0.40
PIK3CG P48736 2/20 0.39
TSHR P16473 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
THRB P10828 1/20 0.37
POLB P06746 2/20 0.37
TP53 P04637 2/20 0.36
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CHRM1 P11229 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923825 1.00 REN (0.42) RENMAPTCYP3A4SMPD1PIK3CG
SCHEMBL2914734 0.86 TSHR (0.40) RENMAPTCYP3A4SMPD1PIK3CG
SCHEMBL2924802 0.86 TSHR (0.40) RENMAPTCYP3A4SMPD1PIK3CG
SCHEMBL3464412 0.86 REN (0.37) RENMAPTCYP3A4THRBCYP2D6
SCHEMBL2923764 0.86 REN (0.37) RENMAPTCYP3A4THRBCYP2D6
SCHEMBL8466898 0.85 REN (0.52) RENCYP3A4
SCHEMBL3557454 0.84 REN (0.34) RENMAPTCYP3A4POLBCYP2C19
SCHEMBL3553031 0.83 REN (0.41) RENMAPTCYP3A4SMPD1PIK3CG
SCHEMBL2921036 0.82 REN (0.42) RENMAPTCYP3A4SMPD1PIK3CG
SCHEMBL4647385 0.81 MAPT (0.41) RENMAPTCYP3A4SMPD1PIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863803-A2 SUBSTITUTED PIPERIDINES Speedel Experimenta AG (CH) 2007-12-12 EP disclosed
WO-2006103277-A2 2 , 4 , 5-SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS SPEEDEL EXPERIMENTA AG (CH) 2006-10-05 WO disclosed