SCHEMBL4647385

SCHEMBL4647385

COCCCN1C(=O)COc2ccc(CO[C@H]3CN(C(=O)O)[C@@H](C(=O)O)C[C@@H]3c3ccc(OC)cc3)cc21

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.41
TSHR P16473 1/20 0.40
SMPD1 P17405 1/20 0.39
REN P00797 3/20 0.38
THRB P10828 1/20 0.38
POLB P06746 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PIK3CG P48736 1/20 0.37
TP53 P04637 2/20 0.37
CYP3A4 P08684 1/20 0.37
CHRM1 P11229 1/20 0.35
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4646330 0.91 MAPT (0.41) MAPTTSHRSMPD1RENTHRB
SCHEMBL5503959 0.87 REN (0.36) MAPTRENTHRBCYP3A4ALDH1A1
SCHEMBL2925488 0.85 MAPT (0.40) MAPTTSHRSMPD1RENL3MBTL1
SCHEMBL4136437 0.85 MAPT (0.42) MAPTTSHRSMPD1RENTHRB
SCHEMBL2921432 0.84 TSHR (0.39) MAPTTSHRSMPD1RENTHRB
SCHEMBL5507277 0.81 REN (0.36) MAPTRENTHRBCYP3A4ALDH1A1
SCHEMBL3906082 0.81 MAPT (0.42) MAPTTSHRSMPD1RENTHRB
SCHEMBL2923825 0.81 REN (0.42) MAPTTSHRSMPD1RENTHRB
SCHEMBL5509732 0.81 REN (0.42) MAPTTSHRSMPD1RENTHRB
SCHEMBL1036573 0.80 MAPT (0.41) MAPTTSHRSMPD1RENTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1958634-A2 Substituted piperidines as inhibitors of beta-secretase, cathepsin D, plasmepsin II and/or HIV protease Speedel Experimenta AG (CH) 2008-08-20 EP disclosed