SCHEMBL5510227

SCHEMBL5510227

N#Cc1ccc2nccc(OCC3C4CNCC43)c2c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 8/20 0.51
GAK O14976 1/20 0.41
RIPK2 O43353 1/20 0.41
COQ8A Q8NI60 1/20 0.41
NLK Q9UBE8 1/20 0.41
CCNC P24863 1/20 0.40
CDK8 P49336 1/20 0.40
SSTR4 P31391 2/20 0.39
PDE5A O76074 1/20 0.39
SLC22A12 Q96S37 1/20 0.38
PDPK1 O15530 3/20 0.38
AR P10275 1/20 0.37
IDO1 P14902 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5510222 1.00 IRAK4 (0.51) IRAK4GAKRIPK2COQ8ANLK
Hydrochloric Acid SCHEMBL23699139 0.81 IRAK4 (0.52) IRAK4SSTR4IDO1
Hydrochloric Acid SCHEMBL30444717 0.81 IRAK4 (0.52) IRAK4SSTR4IDO1
SCHEMBL24010750 0.74 GAK (0.64) GAKRIPK2COQ8ANLKCCNC
SCHEMBL3254205 0.73 SLC22A12 (0.45) IRAK4CCNCCDK8SLC22A12AR
SCHEMBL3254209 0.73 SLC22A12 (0.45) IRAK4CCNCCDK8SLC22A12AR
SCHEMBL23999791 0.73 GAK (0.49) IRAK4GAKRIPK2COQ8ANLK
SCHEMBL4659915 0.71 SLC22A12 (0.45) IRAK4GAKRIPK2COQ8ANLK
SCHEMBL14782742 0.70 HSD11B1 (0.44)
SCHEMBL25830886 0.68 GAK (0.46) GAKRIPK2COQ8ANLKCCNC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed