SCHEMBL5511779

SCHEMBL5511779

COC(=O)C1CCC(COc2ncnc3ccc(OC)cc23)N(C(=O)OC(C)(C)C)C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 6/20 0.47
MTNR1A P48039 4/20 0.47
PIK3CD O00329 4/20 0.44
PIK3CA P42336 4/20 0.44
PIK3CB P42338 2/20 0.44
PIK3CG P48736 2/20 0.44
STS P08842 1/20 0.38
ENPP1 P22413 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
ERBB2 P04626 1/20 0.37
BRAF P15056 1/20 0.37
KDR P35968 1/20 0.37
MAPK14 Q16539 1/20 0.37
TNNI3K Q59H18 1/20 0.37
MAPK7 Q13164 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5511774 1.00 MTNR1B (0.47) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL5511776 1.00 MTNR1B (0.47) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL5507684 0.82 CA1 (0.40) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL632999 0.80 PIK3CD (0.51) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL924200 0.77 PIK3CD (0.51) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL5506799 0.77 MTNR1B (0.41) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL632727 0.76 PIK3CD (0.47) MTNR1BMTNR1APIK3CDPIK3CAPIK3CB
SCHEMBL15179604 0.75 EPHX2 (0.42) MTNR1ASTSKDM4ENPC1RAB9A
SCHEMBL27158644 0.73 SMN1; SMN2 (0.38) STSNPC1MEN1ALDH1A1KMT2A
SCHEMBL632811 0.73 PIK3CD (0.76) MTNR1BPIK3CDPIK3CAPIK3CBPIK3CG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed