SCHEMBL5513007

SCHEMBL5513007

CC(C)c1cc(CC(=O)O)n[nH]1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.56
HCAR3 P49019 1/20 0.56
THRA P10827 6/20 0.43
THRB P10828 6/20 0.43
PRKAB2 O43741 5/20 0.40
PRKAG1 P54619 5/20 0.40
PRKAA2 P54646 5/20 0.40
PRKAA1 Q13131 5/20 0.40
PRKAG3 Q9UGI9 5/20 0.40
PRKAG2 Q9UGJ0 5/20 0.40
PRKAB1 Q9Y478 5/20 0.40
CCNA2 P20248 1/20 0.39
CDK2 P24941 1/20 0.39
CCNA1 P78396 1/20 0.39
KDM5A P29375 6/20 0.37
KDM5C P41229 1/20 0.36
KDM5B Q9UGL1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12740609 0.77 HCAR2 (0.48) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL877436 0.76 HCAR2 (0.52) HCAR2THRATHRBCCNA2CDK2
SCHEMBL1204783 0.75 HCAR2 (0.46) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
Hydrochloric Acid SCHEMBL1371875 0.74 HCAR2 (0.50) HCAR2THRATHRBCCNA2CDK2
SCHEMBL5989046 0.73 HCAR2 (0.37) HCAR2THRATHRB
SCHEMBL1206441 0.73 HCAR2 (0.44) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL28845246 0.73 HCAR2 (0.44) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL1592992 0.72 GABRA5 (0.43) HCAR2THRATHRB
SCHEMBL16619358 0.72 HCAR2 (0.43) HCAR2HCAR3PRKAB2PRKAG1PRKAA2
SCHEMBL1739326 0.72 HCAR2 (1.00) HCAR2HCAR3KDM5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8367666-B2 3-carbamoyl-2-pyridone derivatives SHIONOGI & CO., LTD. (JP) 2013-02-05 US disclosed
US-8178681-B2 methyl 3-methyl-2-{[2-oxo-1-(2-oxo-ethyl)-1,2,5,6,7,8,9,10-octahydro-cycloocta[b]pyridine-3-carbonyl]-amino}-butyrate; cannabinoid receptor agonist; antiinflammatory agent, immunostimulant, analgesic; atopic dermatitis; excellent in photostability, and have excellent transdermal and oral absorbency SHIONOGI & CO., LTD. (JP) 2012-05-15 US disclosed