SCHEMBL5513396

SCHEMBL5513396

CC(C)(C)OC(=O)c1c(-c2cc(C(F)(F)F)cc(S(=O)(=O)NC3CCCCC3)c2)[nH]c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
MAPT P10636 3/20 0.40
LMNA P02545 3/20 0.40
TP53 P04637 2/20 0.40
STS P08842 1/20 0.39
KMT2A Q03164 2/20 0.38
ALDH1A1 P00352 1/20 0.38
PDK1 Q15118 1/20 0.38
PDK2 Q15119 1/20 0.38
PDK3 Q15120 1/20 0.38
PDK4 Q16654 1/20 0.38
MAP2K4 P45985 1/20 0.38
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
IDH2 P48735 2/20 0.37
GABRP O00591 1/20 0.37
GABRD O14764 1/20 0.37
GABRA1 P14867 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5621435 0.87 TDP1 (0.41) TDP1MAPTLMNATP53KMT2A
SCHEMBL5510395 0.86 MEN1 (0.46) TDP1LMNAKMT2AALDH1A1GAA
SCHEMBL5509703 0.83 GLA (0.43) TDP1MAPTLMNATP53STS
SCHEMBL5509086 0.81 BRD4 (0.48) NR1H2TDP1MAPTLMNATP53
SCHEMBL5514925 0.81 MAPT (0.41) TDP1MAPTLMNATP53ALDH1A1
SCHEMBL27720095 0.81 MAPT (0.40) TDP1MAPTLMNATP53KMT2A
SCHEMBL5516306 0.81 ALDH1A1 (0.44) NR1H2TDP1LMNATP53KMT2A
SCHEMBL3996870 0.81 BRD4 (0.47) NR1H2TDP1LMNATP53KMT2A
SCHEMBL5507312 0.80 BRD4 (0.51) TP53GAAHTTBRD4
Tert-Butyl Formate SCHEMBL27720068 0.75 BRD4 (0.38) NR1H2TDP1MAPTLMNATP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1844011-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS Aventis Pharmaceuticals Inc. (US) 2007-10-17 EP disclosed
WO-2006081343-A1 2-PHENYL-INDOLES AS PROSTAGLANDIN D2 RECEPTOR ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2006-08-03 WO disclosed