SCHEMBL5515065

SCHEMBL5515065

COc1ccc(C(=O)C=Cc2ccc(O)cc2)c(O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABCG2 Q9UNQ0 7/20 0.91
MAPT P10636 5/20 0.91
APP P05067 5/20 0.91
LMNA P02545 4/20 0.91
MEN1 O00255 4/20 0.91
MAPK1 P28482 4/20 0.91
KMT2A Q03164 4/20 0.91
CYP3A4 P08684 4/20 0.91
CYP2C19 P33261 3/20 0.91
SMN1; SMN2 Q16637 2/20 0.91
HPGD P15428 3/20 0.86
ALOX15 P16050 3/20 0.86
HSD17B10 Q99714 3/20 0.86
ALDH1A1 P00352 2/20 0.86
TP53 P04637 2/20 0.86
MAOB P27338 2/20 0.82
CTSL P07711 1/20 0.82
NPC1 O15118 1/20 0.82
RECQL P46063 1/20 0.82
RAB9A P51151 1/20 0.82

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30383218 1.00 ABCG2 (0.91) ABCG2MAPTAPPLMNAMEN1
SCHEMBL5515061 1.00 ABCG2 (0.91) ABCG2MAPTAPPLMNAMEN1
SCHEMBL25188859 0.97 ABCG2 (0.97) ABCG2MAPTAPPLMNAMEN1
SCHEMBL30382670 0.95 ABCG2 (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL30384538 0.95 ABCG2 (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL634186 0.95 ABCG2 (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL634187 0.95 ABCG2 (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL25189208 0.95 ABCG2 (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL25219780 0.93 MAPT (1.00) ABCG2MAPTAPPLMNAMEN1
SCHEMBL633177 0.93 MAPT (1.00) ABCG2MAPTAPPLMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3562803-B1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA UNIV DEGLI STUDI ROMA LA SAPIENZA (IT) 2025-10-15 EP claimed
US-20210363121-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA UNIV DEGLI STUDI ROMA LA SAPIENZA (IT) 2021-11-25 US claimed
US-20190337916-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA FONDAZIONE ISTITUTO ITALIANO DI TECNOLOGIA (IT) 2019-11-07 US claimed
US-20070092551-A1 Therapeutic agent TAKARA BIO INC. (JP) 2007-04-26 US claimed
EP-1623704-A1 THERAPEUTIC AGENT TAKARA BIO INC. (JP) 2006-02-08 EP claimed
US-20210363121-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA UNIV DEGLI STUDI ROMA LA SAPIENZA (IT) 2021-11-25 US disclosed
US-20190337916-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA FONDAZIONE ISTITUTO ITALIANO DI TECNOLOGIA (IT) 2019-11-07 US disclosed
US-20070092551-A1 Therapeutic agent TAKARA BIO INC. (JP) 2007-04-26 US disclosed
EP-1623704-A1 THERAPEUTIC AGENT TAKARA BIO INC. (JP) 2006-02-08 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190337916-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA NOTCH1, DNER, NOTCH2 ABCG2 2354/4885MAPT 4067/4885APP 462/4885
US-20070092551-A1 Therapeutic agent FABP4, GPR119, IAPP ABCG2 806/4885MAPT 2256/4885APP 1333/4885
US-20210363121-A1 NOTCH INHIBITORS FOR USE IN THE TREATMENT OF T-CELL ACUTE LYMPHOBLASTIC LEUKEMIA NOTCH1, DNER, NOTCH2 ABCG2 2354/4885MAPT 4067/4885APP 462/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.