SCHEMBL5526262

SCHEMBL5526262

O=C(O)c1cc(-c2ccc(Cl)cn2)n(-c2ccccn2)n1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
MARS1 P56192 6/20 0.63
L3MBTL1 Q9Y468 1/20 0.49
RPA1 P27694 5/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
PPP1CA P62136 3/20 0.44
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
ATM Q13315 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27668789 0.87 MARS1 (0.53) MARS1L3MBTL1RPA1PPP1CAKMT2A
SCHEMBL4927931 0.86 MARS1 (0.52) MARS1RPA1SMN1; SMN2PPP1CAKMT2A
SCHEMBL5521156 0.84 ALDH1A1 (0.52) MARS1SMN1; SMN2KMT2AMEN1
SCHEMBL5524835 0.84 CNR1 (0.50) MARS1KMT2AMEN1
SCHEMBL5522350 0.84 MARS1 (0.50) MARS1L3MBTL1RPA1PPP1CAKMT2A
SCHEMBL27619816 0.81 RPA1 (0.45) MARS1L3MBTL1RPA1SMN1; SMN2PPP1CA
SCHEMBL27668657 0.80 MDM2 (0.56) MARS1
SCHEMBL4932725 0.80 MARS1 (0.64) MARS1L3MBTL1RPA1SMN1; SMN2PPP1CA
SCHEMBL2916915 0.79 MARS1 (0.49) MARS1L3MBTL1RPA1SMN1; SMN2PPP1CA
SCHEMBL5978029 0.79 MARS1 (0.46) MARS1RPA1PPP1CAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070219210-A1 Amidopyrazole Derivative DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-09-20 US disclosed
US-20070219210-A1 Amidopyrazole Derivative DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-09-20 US disclosed
US-20070219210-A1 Amidopyrazole Derivative DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2007-09-20 US disclosed
CN-1902191-A Amidopyrazole derivative DAIICHI SEIYAKU CO (JP) 2007-01-24 CN disclosed
EP-1698626-A1 AMIDOPYRAZOLE DERIVATIVE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2006-09-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070219210-A1 Amidopyrazole Derivative PTGER1, PTGS1, PTGER2 MARS1 2982/4885L3MBTL1 3071/4885RPA1 1661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.