SCHEMBL5528686

SCHEMBL5528686

CNc1nc(N)nc2cc(-c3c(OCCOC)cccc3C(F)(F)F)ccc12.CNc1nc(N)nc2cc(-c3cc(F)c(OC)c(OCCOC)c3)ccc12

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 10/20 0.47
TRPV1 Q8NER1 4/20 0.36
CYBB P04839 1/20 0.35
NCF1 P14598 1/20 0.35
PIK3CA P42336 1/20 0.33
DHFR P00374 1/20 0.33
RAF1 P04049 1/20 0.33
BRAF P15056 1/20 0.33
LRRK2 Q5S007 1/20 0.33
AR P10275 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4524484 0.91 PTPN1 (0.52) PTPN1TRPV1DHFRAR
SCHEMBL4529999 0.88 PIK3CA (0.37) PTPN1CYBBNCF1PIK3CADHFR
SCHEMBL5498432 0.83 PTPN1 (0.51) PTPN1TRPV1DHFR
SCHEMBL4523462 0.83 PTPN1 (0.51) PTPN1TRPV1DHFR
SCHEMBL4524961 0.81 PTPN1 (0.52) PTPN1TRPV1DHFR
SCHEMBL4523940 0.77 PTPN1 (0.64) PTPN1
SCHEMBL4527944 0.77 PTPN1 (0.57) PTPN1TRPV1DHFR
SCHEMBL4528751 0.76 DHFR (0.39) PTPN1PIK3CADHFR
SCHEMBL4520756 0.76 PTPN1 (0.47) PTPN1TRPV1DHFR
Trifluoroacetic Acid SCHEMBL4534719 0.76 PTPN1 (0.47) PTPN1TRPV1DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1812409-A1 AMINOQUINAZOLINES COMPOUNDS F. Hoffmann-Roche AG (CH) 2007-08-01 EP disclosed
WO-2006050843-A1 AMINOQUINAZOLINES COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2006-05-18 WO disclosed