SCHEMBL5532807

SCHEMBL5532807

OCC1NCCc2c1[nH]c1ccccc21

nearest known ligand 0.70

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 1/20 0.70
HTR7 P34969 8/20 0.60
CYP3A4 P08684 1/20 0.60
CYP2D6 P10635 1/20 0.60
CYP2C19 P33261 1/20 0.60
CHRM4 P08173 5/20 0.60
CTSK P43235 1/20 0.60
MAPKAPK2 P49137 1/20 0.59
DRD2 P14416 3/20 0.58
HTR2A P28223 3/20 0.54
HTR2C P28335 3/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29756361 0.85 GRIN2B (0.70) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL10924004 0.85 GRIN2B (0.70) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL21883968 0.85 GRIN2B (0.70) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL8322968 0.85 GRIN2B (0.70) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL3246180 0.83 GRIN2B (0.67) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
Fenharmane SCHEMBL9695673 0.82 GRIN2B (1.00) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
Fenharmane SCHEMBL9696484 0.81 GRIN2B (0.97) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL34463426 0.81 GRIN2B (0.65) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
SCHEMBL18669422 0.81 GRIN2B (0.65) GRIN2BHTR7CYP3A4CYP2D6CYP2C19
Xestoamine SCHEMBL2271935 0.81 GRIN2B (0.65) GRIN2BHTR7CYP3A4CYP2D6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007147819-A1 3H,11H-OXAZOLO[3',4':1,2]PYRIDO[3,4-B]INDOLE DERIVATIVES AND THERAPEUTIC USE THEREOF FOURTILLAN (FR) 2007-12-27 WO disclosed
US-4625032-A LIVER DISORDERS TANABE SEIYAKU CO., LTD. (JP) 1986-11-25 US disclosed
EP-0165017-A2 Novel tetrahydro-B-carboline derivative and processes for preparation thereof Tanabe Seiyaku Co., Ltd. (JP) 1985-12-18 EP disclosed