SCHEMBL5536636

SCHEMBL5536636

CC1(CN2CCOC2=O)CO1

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 2/20 0.40
KDM4E B2RXH2 1/20 0.37
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
NAAA Q02083 1/20 0.33
NQO2 P16083 1/20 0.32
PER2 O15055 1/20 0.31
CRY2 Q49AN0 1/20 0.31
GRM2 Q14416 1/20 0.31
PARG Q86W56 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30047361 0.71 KDM4E (0.42) PIK3CDKDM4ECNR1CNR2NAAA
SCHEMBL261199 0.71
SCHEMBL11983582 0.69 PIK3CD (0.42) PIK3CDKDM4ECNR1CNR2NAAA
SCHEMBL8593693 0.69
SCHEMBL9623993 0.68 PIK3CD (0.44) PIK3CDKDM4ECNR1CNR2NAAA
SCHEMBL2781821 0.68
SCHEMBL11062023 0.68 PIK3CD (0.46) PIK3CDKDM4ECNR1CNR2NAAA
SCHEMBL631171 0.68 PIK3CD (0.41) PIK3CDKDM4ECNR1CNR2NAAA
SCHEMBL17138490 0.68 PER2 (0.36) PER2CRY2
SCHEMBL6153134 0.67 TP53 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2570418-A2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles compound OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2013-03-20 EP disclosed
EP-1555267-B1 2,3-DIHYDRO-6-NITROIMIDAZO[2,1-b]OXAZOLES OTSUKA PHARMA CO LTD (JP) 2013-01-16 EP disclosed
US-7262212-B2 2,3-dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-08-28 US disclosed
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2006-05-04 US disclosed
EP-1555267-A1 2,3-DIHYDRO-6-NITROIMIDAZO 2,1-b OXAZOLES OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2005-07-20 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060094767-A1 2,3-Dihydro-6-nitroimidazo[2,1-b]oxazoles NR2C2, NR4A3, NR4A2 PIK3CD 4528/4885KDM4E 4854/4885CNR1 857/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.