SCHEMBL5540176

SCHEMBL5540176

COC(=O)CCCn1c(=O)n(CC(=O)OC(C)(C)C)c2cccc([N+](=O)[O-])c21.[NaH]

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.39
ALDH1A1 P00352 3/20 0.38
KDM4E B2RXH2 2/20 0.38
NPC1 O15118 1/20 0.37
GAA P10253 1/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
CNR2 P34972 7/20 0.35
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
MAPT P10636 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
PSEN1 P49768 1/20 0.33
PSEN2 P49810 1/20 0.33
APH1B Q8WW43 1/20 0.33
NCSTN Q92542 1/20 0.33
APH1A Q96BI3 1/20 0.33
PSENEN Q9NZ42 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL259712 0.99 LMNA (0.39) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL5540182 0.97 LMNA (0.38) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL2054568 0.91 KDM4E (0.43) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL261021 0.84 ALDH1A1 (0.43) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL260808 0.84 KDM4E (0.50) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL261770 0.83 KDM4E (0.41) ALDH1A1KDM4ENPC1GAASMN1; SMN2
SCHEMBL14538682 0.74 KDM4E (0.47) LMNAALDH1A1KDM4ENPC1GAA
SCHEMBL260929 0.72 APEX1 (0.57) KDM4ENPC1GAAMEN1KMT2A
SCHEMBL260928 0.72 APEX1 (0.57) KDM4ENPC1GAAMEN1KMT2A
SCHEMBL18171837 0.71 ALDH1A1 (0.49) ALDH1A1KDM4ENPC1GAASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1794146-A2 TRICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS Merck & Co., Inc. (US) 2007-06-13 EP disclosed
WO-2006031676-A2 TRICYCLIC ANILIDE SPIROHYDANTOIN CGRP RECEPTOR ANTAGONISTS MERCK & CO., INC. (US) 2006-03-23 WO disclosed