SCHEMBL5540308

SCHEMBL5540308

O=C(NC1N=CC2=CN(S(=O)(=O)c3cccs3)CCC2=N1)c1ccc(F)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
HTR2A P28223 1/20 0.36
POLB P06746 3/20 0.34
MAPT P10636 2/20 0.34
RORC P51449 1/20 0.34
RECQL P46063 1/20 0.34
MCHR1 Q99705 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 1/20 0.33
EPHX2 P34913 1/20 0.33
MKNK1 Q9BUB5 1/20 0.32
SLC6A9 P48067 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540316 0.75 MAPT (0.39) POLBMAPTRORCSMN1; SMN2ALDH1A1
SCHEMBL5540826 0.74 KMT2A (0.44) MAPTRORCSMN1; SMN2ALDH1A1LMNA
SCHEMBL3531915 0.62 MAPK1 (0.44) POLBMAPTRORCSMN1; SMN2ALDH1A1
SCHEMBL7153163 0.58 MEN1 (0.51) POLBMAPTRECQLSMN1; SMN2ALDH1A1
SCHEMBL531986 0.56 MCHR1 (0.64) MCHR1SMN1; SMN2NPC1RAB9A
SCHEMBL24359908 0.54 MCHR1 (0.60) MCHR1NPC1RAB9A
SCHEMBL3282365 0.54 TSHR (0.67) SMN1; SMN2ALDH1A1
SCHEMBL7226660 0.53 POLB (0.62) POLBALDH1A1NPC1RAB9A
SCHEMBL7226664 0.53 POLB (0.62) POLBALDH1A1NPC1RAB9A
SCHEMBL30940072 0.53 HPGDS (0.58) MAPTSMN1; SMN2ALDH1A1LMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed