SCHEMBL5541223

SCHEMBL5541223

CCOC(=O)c1cn2c3c(c(F)c(F)cc3c1=O)OCC2C

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 3/20 0.55
TOP2B Q02880 3/20 0.55
KDM4E B2RXH2 5/20 0.55
KMT2A Q03164 1/20 0.55
CNR1 P21554 1/20 0.54
CNR2 P34972 1/20 0.54
ALDH1A1 P00352 4/20 0.54
HPGD P15428 4/20 0.54
HSD17B10 Q99714 2/20 0.54
ALB P02768 1/20 0.54
HRH3 Q9Y5N1 1/20 0.54
TUBB4A P04350 4/20 0.53
TUBB P07437 4/20 0.53
TUBA3C P0DPH7 4/20 0.53
TUBA1B P68363 4/20 0.53
TUBA4A P68366 4/20 0.53
TUBB4B P68371 4/20 0.53
TUBB3 Q13509 4/20 0.53
TUBB2A Q13885 4/20 0.53
TUBB8 Q3ZCM7 4/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30306119 1.00 TOP2A (0.55) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL2339241 1.00 TOP2A (0.55) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL20125115 0.92 TOP2A (0.55) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL19751491 0.92 TOP2A (0.55) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL15828544 0.90 TOP2A (0.54) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL11200216 0.90 TOP2A (0.49) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL10835611 0.90 TOP2A (0.54) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL25374200 0.90 CNR2 (0.67) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL30542704 0.90 CNR2 (0.67) TOP2ATOP2BKDM4EKMT2ACNR1
SCHEMBL1344388 0.89 CNR1 (0.58) TOP2ATOP2BKDM4EKMT2ACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-60075489-A None JP disclosed
WO-2023158862-A2 STIMULATOR OF INTERFERON GENES (STING) MODULATORS, AND COMPOSITIONS AND METHODS THEREOF GEODE THERAPEUTICS INC. (US) 2023-08-24 WO disclosed
US-20070244318-A1 Process for the Preparation of Levofloxacin Hemihydrate RAO DAVULURI R 2007-10-18 US disclosed
US-6229017-B1 BY ACYLATION AND CYCLIZATION OF A BENZOYL CHLORIDE OR NICOTINOYL CHLORIDE IN THE PRESENCE OF A NON-POLAR TO SLIGHTLY POLAR SOLVENT WITHOUT SEPARATION OF CHEMICAL INTERMEDIATES DURING PROCESS BAYER AKTIENGESELLSCHAFT (DE) 2001-05-08 US disclosed
EP-0206283-B1 OPTICALLY ACTIVE PYRIDOBENZOXAZINE DERIVATIVES DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1993-01-27 EP disclosed
US-5153203-A QUINOLONE DERIVATIVES AND SALTS THEREOF, PREPARATION PROCESSES THEREOF, AND ANTIBACTERIAL AGENTS CONTAINING THE SAME WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1992-10-06 US disclosed
US-5142046-A Optically active pyridobenzoxazine derivatives and intermediates thereof DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1992-08-25 US disclosed
US-5053407-A OPTICALLY ACTIVE PYRIDOBENZOXAZINE DERIVATIVES AND ANTI-MICROBIAL USE DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1991-10-01 US disclosed
US-4985557-A OFLOXACIN INTERMEDIATE DAIICHI SEIYAKU CO., LTD. (JP) 1991-01-15 US disclosed
EP-0390215-A2 Quinolone derivatives and salts thereof, preparation process es thereof, and antibacterial agents containing the same WAKUNAGA SEIYAKU KABUSHIKI KAISHA (JP) 1990-10-03 EP disclosed
US-4958045-A ENAMINES, BACTERICIDES, ANIMAL GROWTH REGULATORS BAYER AKTIENGESELLSCHAFT (DE) 1990-09-18 US disclosed
US-4859773-A Preparation of 1,8-bridged 4-quinoline-3-carboxylic acids BAYER AKTIENGESELLSCHAFT (DE) 1989-08-22 US disclosed
US-4826985-A Intermediates for preparation of racemate and optically active ofloxacin and related derivatives ABBOTT LABORATORIES (US) 1989-05-02 US disclosed
US-4777253-A Process for preparation of racemate and optically active ofloxacin and related derivatives ABBOTT LABORATORIES (US) 1988-10-11 US disclosed
US-4762831-A PROMOTE ANIMAL GROWTH BAYER AKTIENGESELLSCHAFT (DE) 1988-08-09 US disclosed
JP-S6075489-A BORON CHELATE COMPOUND DAI ICHI SEIYAKU CO LTD 1985-04-27 JP disclosed
EP-0047005-B1 BENZOXAZINE DERIVATIVES DAIICHI SEIYAKU CO., LTD. (JP) 1984-11-14 EP disclosed
US-4382892-A Benzoxazine derivatives DAIICHI SEIYAKU CO., LTD. (JP) 1983-05-10 US disclosed
EP-0047005-A1 Benzoxazine derivatives DAIICHI SEIYAKU CO., LTD. (JP) 1982-03-10 EP disclosed
JP-S0675489-A 0001-01-01 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070244318-A1 Process for the Preparation of Levofloxacin Hemihydrate RTF1, CYP2F1, CYP4F11 TOP2A 744/4885TOP2B 1081/4885KDM4E 1527/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.