SCHEMBL5543503

SCHEMBL5543503

CC(C)c1nc(NCCc2cccnc2)c2n[nH]c(=O)n2c1C(O)CCc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.50
GSK3A P49840 4/20 0.40
GSK3B P49841 4/20 0.40
GBA1 P04062 3/20 0.38
F2 P00734 1/20 0.38
PDE5A O76074 2/20 0.37
LMNA P02545 1/20 0.36
CTSL P07711 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
JAK3 P52333 1/20 0.35
PDE9A O76083 1/20 0.34
CSNK2A2 P19784 1/20 0.34
CSNK2B P67870 1/20 0.34
CSNK2A1 P68400 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543633 0.94 ADORA1 (0.50) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5550010 0.90 ADORA1 (0.45) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5545500 0.88 ADORA1 (0.49) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549322 0.85 ADORA1 (0.45) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549074 0.84 ADORA1 (0.49) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5548924 0.84 ADORA1 (0.54) ADORA1GSK3AGSK3BGBA1PDE5A
SCHEMBL5543764 0.83 ADORA1 (0.43) ADORA1CYP1A2CYP3A4CYP2C19
SCHEMBL3525903 0.83 ADORA1 (0.50) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549397 0.82 ADORA1 (0.43) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5543583 0.82 ADORA1 (0.43) ADORA1GSK3AGSK3BF2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed