SCHEMBL5545500

SCHEMBL5545500

CC(C)(C)c1nc(NCCc2cccnc2)c2n[nH]c(=O)n2c1C(O)CCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.49
GSK3A P49840 4/20 0.39
GSK3B P49841 4/20 0.39
GBA1 P04062 3/20 0.38
F2 P00734 1/20 0.38
PDE5A O76074 2/20 0.36
CTSL P07711 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
JAK3 P52333 1/20 0.34
LMNA P02545 2/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5549322 0.97 ADORA1 (0.45) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549074 0.96 ADORA1 (0.49) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5543583 0.94 ADORA1 (0.43) ADORA1GSK3AGSK3BF2JAK3
SCHEMBL5549397 0.94 ADORA1 (0.43) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5548564 0.92 ADORA1 (0.42) ADORA1GSK3AGSK3BCYP3A4CYP2D6
SCHEMBL3525368 0.89 ADORA1 (0.44) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5543503 0.88 ADORA1 (0.50) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5548882 0.87 ADORA1 (0.45) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5545565 0.83 ADORA1 (0.42) ADORA1CYP1A2CYP3A4CYP2C19MEN1
SCHEMBL5548920 0.82 ADORA1 (0.50) ADORA1GSK3AGSK3BGBA1F2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed