SCHEMBL5548924

SCHEMBL5548924

CC(C)c1nc(NCCc2cccnc2)c2n[nH]c(=O)n2c1-c1ccccc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.54
GBA1 P04062 7/20 0.48
PDE5A O76074 4/20 0.44
GSK3A P49840 4/20 0.42
GSK3B P49841 4/20 0.42
ALDH1A1 P00352 3/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C19 P33261 2/20 0.39
POLB P06746 1/20 0.39
CYP2C9 P11712 1/20 0.39
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3525903 0.87 ADORA1 (0.50) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5543633 0.86 ADORA1 (0.50) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5550083 0.85 ADORA1 (0.53) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5543503 0.84 ADORA1 (0.50) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5550010 0.81 ADORA1 (0.45) ADORA1GBA1GSK3AGSK3BMAPK1
SCHEMBL5549306 0.79 ADORA1 (0.52) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5548429 0.79 ADORA1 (0.53) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL3527078 0.77 ADORA1 (0.46) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5548920 0.76 ADORA1 (0.50) ADORA1GBA1PDE5AGSK3AGSK3B
SCHEMBL5543566 0.75 MAPK1 (0.52) ALDH1A1POLBNPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed