SCHEMBL5545002

SCHEMBL5545002

Cc1ccc(CNc2nc(C(C)(C)C)cn3c(=O)[nH]nc23)cn1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 14/20 0.51
GSK3B P49841 14/20 0.51
PDE10A Q9Y233 1/20 0.38
ADORA1 P30542 1/20 0.36
CDK2 P24941 1/20 0.36
CDK9 P50750 1/20 0.36
TLR7 Q9NYK1 2/20 0.36
VNN1 O95497 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3526786 0.91 GSK3B (0.56) GSK3AGSK3BADORA1
SCHEMBL3523080 0.85 GSK3A (0.50) GSK3AGSK3BADORA1
SCHEMBL5548604 0.83 GSK3A (0.48) GSK3AGSK3B
SCHEMBL3528837 0.82 GSK3B (0.47) GSK3AGSK3BADORA1CDK2
SCHEMBL5550039 0.82 GSK3A (0.46) GSK3AGSK3BADORA1CDK2
SCHEMBL5549249 0.81 CA1 (0.46)
SCHEMBL5545469 0.81 ADORA1 (0.41) GSK3AGSK3BADORA1
SCHEMBL5543587 0.81 GSK3B (0.39) GSK3AGSK3BADORA1
SCHEMBL5549013 0.81 ALPL (0.41) GSK3AGSK3BADORA1
SCHEMBL5549004 0.81 PDE10A (0.39) GSK3AGSK3BPDE10AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed