SCHEMBL5548920

SCHEMBL5548920

Cc1c(C(C)(C)C)nc(NCCc2cccnc2)c2n[nH]c(=O)n12

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.50
GSK3A P49840 4/20 0.47
GSK3B P49841 4/20 0.47
INSR P06213 1/20 0.40
IGF1R P08069 1/20 0.40
FGFR1 P11362 1/20 0.40
KDR P35968 1/20 0.40
GBA1 P04062 2/20 0.39
F2 P00734 2/20 0.37
JAK2 O60674 1/20 0.37
PTK2 Q05397 1/20 0.37
PDE4A P27815 1/20 0.37
PDE4B Q07343 1/20 0.37
PDE4C Q08493 1/20 0.37
PDE4D Q08499 1/20 0.37
PRSS1 P07477 1/20 0.37
PDE5A O76074 2/20 0.36
JAK3 P52333 1/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548429 0.88 ADORA1 (0.53) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL3527078 0.85 ADORA1 (0.46) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL5549322 0.85 ADORA1 (0.45) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL5548882 0.85 ADORA1 (0.45) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL3525903 0.84 ADORA1 (0.50) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL3525368 0.83 ADORA1 (0.44) ADORA1GSK3AGSK3BINSRIGF1R
SCHEMBL5545500 0.82 ADORA1 (0.49) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549074 0.82 ADORA1 (0.49) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5549397 0.80 ADORA1 (0.43) ADORA1GSK3AGSK3BGBA1F2
SCHEMBL5543583 0.80 ADORA1 (0.43) ADORA1GSK3AGSK3BF2JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed