SCHEMBL5545525

SCHEMBL5545525

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCc2ccc(Oc3ccccc3)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 2/20 0.47
GSK3B P49841 10/20 0.40
GSK3A P49840 9/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
FES P07332 1/20 0.39
FGFR1 P11362 1/20 0.39
FLT4 P35916 1/20 0.39
KDR P35968 1/20 0.39
EPHX2 P34913 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
DAO P14920 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543493 0.85 GSK3B (0.50) ADORA1GSK3BGSK3A
SCHEMBL5549402 0.85 ADORA1 (0.43) ADORA1GSK3BGSK3A
SCHEMBL5545556 0.85 GSK3A (0.48) ADORA1GSK3BGSK3A
SCHEMBL5548893 0.84 GSK3A (0.49) ADORA1GSK3BGSK3A
SCHEMBL3528033 0.84 GSK3B (0.56) ADORA1GSK3BGSK3A
SCHEMBL5549283 0.84 GSK3B (0.58) ADORA1GSK3BGSK3A
SCHEMBL5549014 0.82 CA1 (0.49) ADORA1CA1CA2CA9
SCHEMBL5550039 0.80 GSK3A (0.46) ADORA1GSK3BGSK3A
SCHEMBL5543514 0.79 GSK3B (0.40) ADORA1GSK3BGSK3A
SCHEMBL5545517 0.79 GSK3B (0.54) ADORA1GSK3BGSK3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed