SCHEMBL5543493

SCHEMBL5543493

CC(C)(C)c1cn2c(=O)[nH]nc2c(NCCc2ccc(Cl)cc2)n1

nearest known ligand 0.50

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.50
GSK3A P49840 14/20 0.44
ADORA1 P30542 1/20 0.43
RXFP1 Q9HBX9 2/20 0.42
TP53 P04637 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
GPR84 Q9NQS5 1/20 0.41
AURKB Q96GD4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5543524 0.89 ADORA1 (0.43) GSK3BGSK3AADORA1GPR84
SCHEMBL5549402 0.89 ADORA1 (0.43) GSK3BGSK3AADORA1MAPTGPR84
SCHEMBL3528033 0.88 GSK3B (0.56) GSK3BGSK3AADORA1
SCHEMBL5545429 0.88 GSK3B (0.46) GSK3BGSK3AADORA1TP53MAPT
SCHEMBL5549014 0.87 CA1 (0.49) ADORA1RXFP1SMN1; SMN2
SCHEMBL5545525 0.85 ADORA1 (0.47) GSK3BGSK3AADORA1
SCHEMBL3526786 0.85 GSK3B (0.56) GSK3BGSK3AADORA1
SCHEMBL5549261 0.84 KMT2A (0.48) RXFP1TP53MAPTSMN1; SMN2
SCHEMBL5545556 0.83 GSK3A (0.48) GSK3BGSK3AADORA1
SCHEMBL3525610 0.82 GSK3B (0.55) GSK3BGSK3AADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed