SCHEMBL5546641

SCHEMBL5546641

CC(C)(C)OC(=O)NCCCCN(Cc1ccc(C(=O)N(Cc2nccn2COCC[Si](C)(C)C)Cc2nccn2COCC[Si](C)(C)C)cc1)C(=O)O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SUCNR1 Q9BXA5 4/20 0.34
CKS1B P61024 1/20 0.34
SKP1 P63208 1/20 0.34
SKP2 Q13309 1/20 0.34
NAMPT P43490 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
CA1 P00915 4/20 0.33
CA2 P00918 4/20 0.33
CA12 O43570 3/20 0.33
CA9 Q16790 3/20 0.33
HDAC3 O15379 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
NCOR2 Q9Y618 1/20 0.33
P2RY14 Q15391 1/20 0.33
MIF P14174 1/20 0.33
CYP3A4 P08684 1/20 0.33
MC4R P32245 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1792634 0.91 MAPT (0.38) CKS1BSKP1SKP2NAMPTMEN1
SCHEMBL1792636 0.85 ATM (0.37) MEN1KMT2ACYP3A4
SCHEMBL1793874 0.78 CXCR4 (0.58) CXCR4
SCHEMBL1796431 0.76 DGAT1 (0.36) MC4R
SCHEMBL1793865 0.75 KMT2A (0.37) MEN1KMT2A
SCHEMBL1797293 0.75 ALDH1A1 (0.39) CXCR4
SCHEMBL1796181 0.75 CXCR4 (0.38) CXCR4
SCHEMBL6749699 0.74 KDM4E (0.44) NAMPTCA1CA2CA12CA9
SCHEMBL3843734 0.73 SUCNR1 (0.37) SUCNR1CKS1BSKP1SKP2MEN1
SCHEMBL5767975 0.72 SSTR4 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1790639-B1 SPIROCYCLIC COMPOUNDS AND THEIR USE AS CXCR4-ANTAGONISTS ONO PHARMACEUTICAL CO (JP) 2014-03-26 EP disclosed
EP-1790639-A1 COMPOUND CONTAINING BASIC GROUP AND USE THEREOF ONO PHARMACEUTICAL CO., LTD. (JP) 2007-05-30 EP disclosed