SCHEMBL5547696

SCHEMBL5547696

CN1CCC(CN2CCN(C(=O)CN(c3ccccc3)c3ccccc3)CC2)CC1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 10/20 0.65
CACNA1B Q00975 10/20 0.65
CACNB1 Q02641 10/20 0.65
CACNA1C Q13936 2/20 0.65
MEN1 O00255 2/20 0.45
ALDH1A1 P00352 2/20 0.45
KMT2A Q03164 2/20 0.45
LMNA P02545 1/20 0.45
KDM4E B2RXH2 1/20 0.45
HTT P42858 1/20 0.45
CHRM4 P08173 2/20 0.43
CHRM5 P08912 2/20 0.43
CHRM1 P11229 2/20 0.43
CHRM3 P20309 2/20 0.43
BDKRB1 P46663 1/20 0.41
TACR2 P21452 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6499599 0.87 CACNA2D1 (0.50) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL13701483 0.81 CACNA2D1 (0.73) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL4841732 0.79 ACHE (0.55) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL3861078 0.79 CACNA2D1 (1.00) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
Hydrochloric Acid SCHEMBL6372221 0.79 ACHE (0.54) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL5548264 0.78 CACNA2D1 (0.55) CACNA2D1CACNA1BCACNB1CACNA1CALDH1A1
SCHEMBL4275876 0.76 CACNA2D1 (0.73) CACNA2D1CACNA1BCACNB1CACNA1CCHRM1
SCHEMBL4286091 0.75 CACNA2D1 (0.71) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL4284711 0.75 CACNA2D1 (0.71) CACNA2D1CACNA1BCACNB1CACNA1CMEN1
SCHEMBL8212834 0.74 CACNA2D1 (0.91) CACNA2D1CACNA1BCACNB1CACNA1CLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1745042-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS Neuromed Pharmaceuticals, Ltd. (CA) 2007-01-24 EP claimed
WO-2005097779-A1 DIARYLAMINE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS NEUROMED PHARMACEUTICALS LTD. (CA) 2005-10-20 WO claimed